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TargetSuppressor of tumorigenicity 14 protein [596-855]
LigandBDBM236493
Substrate/Competitorn/a
Meas. Tech.Inhibition Enzymatic Assay
pH7.4±n/a
Temperature298.15±n/a K
Ki 0.088±0.01 nM
Commentsextracted
Citation Richter, MLeduc, RColombo, EMarsault, E Matriptase inhibitors and uses thereof against orthomyxoviridae infections US Patent US9365853 Publication Date 6/14/2016
More Info.:Get all data from this article,  Assay Method
 
Suppressor of tumorigenicity 14 protein [596-855]
Name:Suppressor of tumorigenicity 14 protein [596-855]
Synonyms:Matriptase | PRSS14 | SNC19 | ST14 | ST14_HUMAN | TADG15
Type:Enzyme
Mol. Mass.:28561.29
Organism:Homo sapiens (Human)
Description:amino acids 596-855
Residue:260
Sequence:
GSDEKDCDCGLRSFTRQARVVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAA
HCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALL
ELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTT
CENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNK
PGVYTRLPLFRDWIKENTGV
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  Blast E-value cutoff:
BDBM236493
n/a
NameBDBM236493
Synonyms:US10988505, Comparative #2 | US9365853, 4
TypeSmall organic molecule
Emp. Form.C21H30N8O4S
Mol. Mass.490.579
SMILESC[C@H](NC(=O)[C@@H](N)CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)c1nc2ccccc2s1 |r|
Structure
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