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TargetCannabinoid receptor 1
LigandBDBM239151
Substrate/Competitorn/a
Meas. Tech.Cannabinoid Receptor Binding Assay
Ki>1.0e+4±n/a nM
IC50>1.0e+4±n/a nM
Citation Taher, ATKadry, HHAllarà, MDi Marzo, VAbadi, AHAbouzid, KA Synthesis and binding study of certain 6-arylalkanamides as molecular probes for cannabinoid receptor subtypes. J Enzyme Inhib Med Chem28:436-9 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cannabinoid receptor 1
Name:Cannabinoid receptor 1
Synonyms:CANN6 | CANNABINOID CB1 | CB-R | CB1 | CNR | CNR1 | CNR1_HUMAN | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cannabinoid receptor 1 (brain)
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:52868.96
Organism:Homo sapiens (Human)
Description:P21554
Residue:472
Sequence:
MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNPQLVPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIA
VLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVF
HRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLM
WTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWK
AHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLL
AIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQ
PLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
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  Blast E-value cutoff:
BDBM239151
n/a
NameBDBM239151
Synonyms:(E)-6-(Biphenyl-4-yl)-N-(2-hydroxybutan-2-yl)-4-oxohex-5-enamide (3m)
TypeSmall organic molecule
Emp. Form.C22H25NO3
Mol. Mass.351.4388
SMILESCCC(C)(O)NC(=O)CCC(=O)\C=C\c1ccc(cc1)-c1ccccc1
Structure
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