| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
|---|
| Ligand | BDBM239153 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Cannabinoid Receptor Binding Assay |
|---|
| Ki | >1.0e+4±n/a nM |
|---|
| IC50 | >1.0e+4±n/a nM |
|---|
| Citation |  Taher, AT; Kadry, HH; Allarà, M; Di Marzo, V; Abadi, AH; Abouzid, KA Synthesis and binding study of certain 6-arylalkanamides as molecular probes for cannabinoid receptor subtypes. J Enzyme Inhib Med Chem28:436-9 (2013) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cannabinoid receptor 1 |
|---|
| Name: | Cannabinoid receptor 1 |
|---|
| Synonyms: | CANN6 | CANNABINOID CB1 | CB-R | CB1 | CNR | CNR1 | CNR1_HUMAN | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cannabinoid receptor 1 (brain) |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 52868.96 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P21554 |
|---|
| Residue: | 472 |
|---|
| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNPQLVPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIA
VLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVF
HRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLM
WTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWK
AHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLL
AIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQ
PLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
|
|
|
|---|
| BDBM239153 |
|---|
| n/a |
|---|
| Name | BDBM239153 |
|---|
| Synonyms: | Ethyl 2-(4-(naphthalen-1-ylamino)-4-oxobutanamido)acetate (5b) |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H20N2O4 |
|---|
| Mol. Mass. | 328.3624 |
|---|
| SMILES | CCOC(=O)CNC(=O)CCC(=O)Nc1cccc2ccccc12 |
|---|
| Structure | 
|
|---|
Search and Browse
