| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Parathyroid hormone/parathyroid hormone-related peptide receptor |
|---|
| Ligand | BDBM64567 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | cAMP Assay |
|---|
| pH | 7.4±n/a |
|---|
| EC50 | 3200±n/a nM |
|---|
| Comments | extracted |
|---|
| Citation |  Nishimura, Y; Esaki, T; Tamura, T Hydantoin derivative US Patent US9428505 Publication Date 8/30/2016 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Parathyroid hormone/parathyroid hormone-related peptide receptor |
|---|
| Name: | Parathyroid hormone/parathyroid hormone-related peptide receptor |
|---|
| Synonyms: | PTH1R_RAT | Parathyroid hormone 1 receptor (PTH1R) | Parathyroid hormone/parathyroid hormone-related peptide receptor | Pth1r | Pthr | Pthr1 |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 66273.93 |
|---|
| Organism: | Rattus norvegicus (Rat) |
|---|
| Description: | P25961 |
|---|
| Residue: | 591 |
|---|
| Sequence: | MGAARIAPSLALLLCCPVLSSAYALVDADDVFTKEEQIFLLHRAQAQCDKLLKEVLHTAA
NIMESDKGWTPASTSGKPRKEKASGKFYPESKENKDVPTGSRRRGRPCLPEWDNIVCWPL
GAPGEVVAVPCPDYIYDFNHKGHAYRRCDRNGSWEVVPGHNRTWANYSECLKFMTNETRE
REVFDRLGMIYTVGYSMSLASLTVAVLILAYFRRLHCTRNYIHMHMFLSFMLRAASIFVK
DAVLYSGFTLDEAERLTEEELHIIAQVPPPPAAAAVGYAGCRVAVTFFLYFLATNYYWIL
VEGLYLHSLIFMAFFSEKKYLWGFTIFGWGLPAVFVAVWVGVRATLANTGCWDLSSGHKK
WIIQVPILASVVLNFILFINIIRVLATKLRETNAGRCDTRQQYRKLLRSTLVLVPLFGVH
YTVFMALPYTEVSGTLWQIQMHYEMLFNSFQGFFVAIIYCFCNGEVQAEIRKSWSRWTLA
LDFKRKARSGSSSYSYGPMVSHTSVTNVGPRAGLSLPLSPRLPPATTNGHSQLPGHAKPG
APATETETLPVTMAVPKDDGFLNGSCSGLDEEASGSARPPPLLQEEWETVM
|
|
|
|---|
| BDBM64567 |
|---|
| n/a |
|---|
| Name | BDBM64567 |
|---|
| Synonyms: | US9428505, Compound 11 |
|---|
| Type | n/a |
|---|
| Emp. Form. | C29H30F3N5O6S |
|---|
| Mol. Mass. | 633.639 |
|---|
| SMILES | Cc1cc(cc(C)c1CCS(=O)(=O)N1CCC2(CC1)N=C(NC2=O)c1ccc(OC(F)(F)F)cc1)N1C(=O)NC(=O)C11CC1 |c:21| |
|---|
| Structure | 
|
|---|
Search and Browse
