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TargetSerine/threonine-protein kinase pim-3
LigandBDBM249016
Substrate/Competitorn/a
Meas. Tech.Kinase Binding Assay
pH7.2±n/a
Temperature298.15±n/a K
Ki 0.026±n/a nM
Commentsextracted
Citation Do, SHu, HKolesnikov, ATsui, VHWang, X 5-azaindazole compounds and methods of use US Patent US9434725 Publication Date 9/6/2016
More Info.:Get all data from this article,  Assay Method
 
Serine/threonine-protein kinase pim-3
Name:Serine/threonine-protein kinase pim-3
Synonyms:PIM3 | PIM3_HUMAN | Serine/threonine-protein kinase pim-3 (PIM3)
Type:Protein
Mol. Mass.:35888.19
Organism:Homo sapiens (Human)
Description:Q86V86
Residue:326
Sequence:
MLLSKFGSLAHLCGPGGVDHLPVKILQPAKADKESFEKAYQVGAVLGSGGFGTVYAGSRI
ADGLPVAVKHVVKERVTEWGSLGGATVPLEVVLLRKVGAAGGARGVIRLLDWFERPDGFL
LVLERPEPAQDLFDFITERGALDEPLARRFFAQVLAAVRHCHSCGVVHRDIKDENLLVDL
RSGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSATVWSLGVLLYDMVC
GDIPFEQDEEILRGRLLFRRRVSPECQQLIRWCLSLRPSERPSLDQIAAHPWMLGADGGV
PESCDLRLCTLDPDDVASTTSSSESL
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  Blast E-value cutoff:
BDBM249016
n/a
NameBDBM249016
Synonyms:US9434725, 247
TypeSmall organic molecule
Emp. Form.C20H21N9
Mol. Mass.387.441
SMILESNc1cncc(n1)-c1cc2n(ncc2cn1)-c1cccc(n1)N1CCCNCC1
Structure
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