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TargetRetinol-binding protein 4
LigandBDBM249466
Substrate/Competitorn/a
Meas. Tech.Scintillation Proximity Binding Assay
pH7.4±n/a
Temperature277.15±n/a K
IC50 4.128382±n/a nM
Commentsextracted
Citation Petrukhin, KCioffi, CJohnson, GAllikmets, RFreeman, EChen, PConlon, MZhu, L Substituted 4-phenylpiperidines, their preparation and use US Patent US9434727 Publication Date 9/6/2016
More Info.:Get all data from this article,  Assay Method
 
Retinol-binding protein 4
Name:Retinol-binding protein 4
Synonyms:PRBP | Plasma retinol-binding protein | RBP | RBP4 | RET4_HUMAN | Retinol-binding protein 4 | Retinol-binding protein 4 (RBP4) | spa binding assay for rbp4
Type:Protein
Mol. Mass.:23008.75
Organism:Homo sapiens (Human)
Description:P02753
Residue:201
Sequence:
MKWVWALLLLAALGSGRAERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIV
AEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGND
DHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLA
RQYRLIVHNGYCDGRSERNLL
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  Blast E-value cutoff:
BDBM249466
n/a
NameBDBM249466
Synonyms:US10072016, Compound 65 | US10407433, Compound 65 | US10913746, Compound 65 | US11649240, Compound 65 | US9434727, 65 | US9777010, Compound 65
TypeSmall organic molecule
Emp. Form.C20H15F4N5O
Mol. Mass.417.3596
SMILESFc1cccc(C2CCN(CC2)C(=O)c2nnc3ccc(cn23)C#N)c1C(F)(F)F
Structure
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