| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 5 |
|---|
| Ligand | BDBM251706 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Receptor Assay |
|---|
| Temperature | 310.15±n/a K |
|---|
| IC50 | 17±n/a nM |
|---|
| Comments | extracted |
|---|
| Citation |  Buffham, W; Canning, H; Davenport, R; Farnaby, W; Mack, S; Parmar, A; Wright, S Compounds US Patent US9464060 Publication Date 10/11/2016 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Lysophosphatidic acid receptor 5 |
|---|
| Name: | Lysophosphatidic acid receptor 5 |
|---|
| Synonyms: | GPR92 | GPR93 | LPAR5 | LPAR5_HUMAN | Lysophosphatidic acid receptor 5 | Lysophosphatidic acid receptor 5 (LPA5) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 41372.36 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q9H1C0 |
|---|
| Residue: | 372 |
|---|
| Sequence: | MLANSSSTNSSVLPCPDYRPTHRLHLVVYSLVLAAGLPLNALALWVFLRALRVHSVVSVY
MCNLAASDLLFTLSLPVRLSYYALHHWPFPDLLCQTTGAIFQMNMYGSCIFLMLINVDRY
AAIVHPLRLRHLRRPRVARLLCLGVWALILVFAVPAARVHRPSRCRYRDLEVRLCFESFS
DELWKGRLLPLVLLAEALGFLLPLAAVVYSSGRVFWTLARPDATQSQRRRKTVRLLLANL
VIFLLCFVPYNSTLAVYGLLRSKLVAASVPARDRVRGVLMVMVLLAGANCVLDPLVYYFS
AEGFRNTLRGLGTPHRARTSATNGTRAALAQSERSAVTTDATRPDAASQGLLRPSDSHSL
SSFTQCPQDSAL
|
|
|
|---|
| BDBM251706 |
|---|
| n/a |
|---|
| Name | BDBM251706 |
|---|
| Synonyms: | US10100018, Example 42 | US9464060, 42 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C25H21ClFNO4 |
|---|
| Mol. Mass. | 453.89 |
|---|
| SMILES | OC(=O)c1ccc(CN(CC2CC2)C(=O)c2ccc(Oc3c(F)cccc3Cl)cc2)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
