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Assay Method Information

Assay Name:  ChEMBL_1295165 (CHEMBL3128666)
Description:  Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins followed by PGD2 challenge measured after 60 mins by chemiluminescence assay
Affinity data for this assay
 

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Last update November 1, 2007
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