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Assay Method Information

Assay Name:  ChEMBL_1620896 (CHEMBL3863179)
Description:  Inverse agonist activity at human CB1 receptor transfected in HEK293 cells assessed as increase of forskolin-induced cAMP production incubated for 30 mins followed by d2 labeled cAMP addition measured after 60 mins by HTRF assay
Affinity data for this assay
 

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Last update November 1, 2007
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