Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM142256 (US8933099, 22 | US9951047, Compound (I)) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 4.5 | n/a | n/a | n/a | n/a | n/a | 25 |
Eisai R&D Management Co., Ltd. US Patent | Assay Description In this assay, the inhibitory activity of a test substance against the tyrosine kinase activity of FGFR2 protein is measured.To each well of a flat b... | US Patent US8933099 (2015) BindingDB Entry DOI: 10.7270/Q28S4NMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM142255 (US8933099, 21) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | 25 |
Eisai R&D Management Co., Ltd. US Patent | Assay Description In this assay, the inhibitory activity of a test substance against the tyrosine kinase activity of FGFR2 protein is measured.To each well of a flat b... | US Patent US8933099 (2015) BindingDB Entry DOI: 10.7270/Q28S4NMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM142236 (US8933099, 2) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.40 | n/a | n/a | n/a | n/a | n/a | 25 |
Eisai R&D Management Co., Ltd. US Patent | Assay Description In this assay, the inhibitory activity of a test substance against the tyrosine kinase activity of FGFR2 protein is measured.To each well of a flat b... | US Patent US8933099 (2015) BindingDB Entry DOI: 10.7270/Q28S4NMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50000130 (CHEMBL320550) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 25.2 | n/a | n/a | n/a | n/a | n/a | n/a |
University College Dublin Curated by ChEMBL | Assay Description 24% inhibition of FGF-2 binding to heparin-albumin by ELISA | Bioorg Med Chem Lett 12: 3287-90 (2002) BindingDB Entry DOI: 10.7270/Q2ZP45G2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167952 (1-(4-(3-Methoxyphenyl)piperazin-1-yl)-3-(quinazoli...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 103 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50331095 (CHEMBL1289494 | Tivozanib | US10464902, Tivozanib) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 114 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167953 (1-(4-(4-Methoxyphenyl)piperazin-1-yl)-3-(quinazoli...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 122 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167954 (1-(4-(3-(Trifluoromethyl)phenyl)piperazin-1-yl)-3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 145 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50000128 (CHEMBL113091) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 149 | n/a | n/a | n/a | n/a | n/a | n/a |
University College Dublin Curated by ChEMBL | Assay Description 23% inhibition of FGF-2 binding to heparin-albumin by ELISA | Bioorg Med Chem Lett 12: 3287-90 (2002) BindingDB Entry DOI: 10.7270/Q2ZP45G2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167956 (1-(4-(3,4-Dichlorophenyl)piperazin-1-yl)-3-(quinaz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 178 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167951 (1-(4-(2-Methoxyphenyl)piperazin-1-yl)-3-(quinazoli...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 209 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167957 (1-(4-(2,4-Dimethylphenyl)piperazin-1-yl)-3-(quinaz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 222 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167950 (1-(4-(4-Nitrophenyl)piperazin-1-yl)-3-(quinazolin-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 248 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167945 (1-(4-Phenylpiperazin-1-yl)-3-(quinazolin-4-yloxy)p...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 293 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167949 (1-(4-(4-Fluorophenyl)piperazin-1-yl)-3-(quinazolin...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50421574 (CHEMBL2303729) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | <313 | n/a | n/a | n/a | n/a | n/a | n/a |
University College Dublin Curated by ChEMBL | Assay Description 25% inhibition of FGF-2 binding to heparin-albumin by ELISA | Bioorg Med Chem Lett 12: 3287-90 (2002) BindingDB Entry DOI: 10.7270/Q2ZP45G2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50421574 (CHEMBL2303729) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
University College Dublin Curated by ChEMBL | Assay Description 25% inhibition of FGF-2 binding to heparin-albumin by ELISA | Bioorg Med Chem Lett 12: 3287-90 (2002) BindingDB Entry DOI: 10.7270/Q2ZP45G2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167948 (1-(4-(2-Fluorophenyl)piperazin-1-yl)-3-(quinazolin...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 372 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167955 (1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-3-(quinaz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 398 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167947 (1-(4-(3-Chlorophenyl)piperazin-1-yl)-3-(quinazolin...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 402 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167959 (1-(4-Methylpiperazin-1-yl)-3-(quinazolin-4-yloxy)p...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 419 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167958 (1-(4-Benzylpiperazin-1-yl)-3-(quinazolin-4-yloxy)p...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 444 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167946 (1-(4-(2-Chlorophenyl)piperazin-1-yl)-3-(quinazolin...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 506 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167960 (1-(4-Ethylpiperazin-1-yl)-3-(quinazolin-4-yloxy)pr...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 519 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167961 (1-(Dimethylamino)-3-(quinazolin-4-yloxy)propan-2-o...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 582 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167965 (1-(2-Methyl-1H-imidazol-1-yl)-3-(quinazolin-4-ylox...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 586 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167966 (1-(4-Methyl-1H-imidazol-1-yl)-3-(quinazolin-4-ylox...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 592 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167963 (1-(Piperidin-1-yl)-3-(quinazolin-4-yloxy)propan-2-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 593 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167962 (1-Morpholino-3-(quinazolin-4-yloxy)propan-2-ol (3r...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 602 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM167964 (1-(1H-Imidazol-1-yl)-3-(quinazolin-4-yloxy)propan-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 609 | n/a | n/a | n/a | n/a | 7.2 | 25 |
Nanjing University | Assay Description VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r... | Chem Biol Drug Des 86: 1323-9 (2015) Article DOI: 10.1111/cbdd.12596 BindingDB Entry DOI: 10.7270/Q2GB22TR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50454865 (CHEMBL4209610) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CSIC and Universidad de Sevilla Curated by ChEMBL | Assay Description Inhibition of fluorescein labelled heparin-like hexasaccharide probe binding to recombinant human FGF-2 after 5 mins by fluorescence polarization ass... | Bioorg Med Chem 26: 1076-1085 (2018) Article DOI: 10.1016/j.bmc.2018.01.022 BindingDB Entry DOI: 10.7270/Q2H41V1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50182286 (CHEMBL3819333) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Parma Curated by ChEMBL | Assay Description Inhibition of human recombinant FGF2 assessed as reduction in HSPG/FGF2/FGDR interaction by measuring FGF2 mediated A475-CHO-flg-1A-luc cell to CHO-K... | J Med Chem 59: 4651-63 (2016) Article DOI: 10.1021/acs.jmedchem.5b02021 BindingDB Entry DOI: 10.7270/Q26Q205Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50182285 (CHEMBL3819473) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Parma Curated by ChEMBL | Assay Description Inhibition of human recombinant FGF2 assessed as reduction in HSPG/FGF2/FGDR interaction by measuring FGF2 mediated A475-CHO-flg-1A-luc cell to CHO-K... | J Med Chem 59: 4651-63 (2016) Article DOI: 10.1021/acs.jmedchem.5b02021 BindingDB Entry DOI: 10.7270/Q26Q205Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50260260 (Biotin-Ala-(Arg)9 | CID44576236 | [amino({[(1R,2S,...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to biotinylated FGF2 in CHO cells by flow cytometry | J Biol Chem 282: 13585-91 (2007) Article DOI: 10.1074/jbc.M700463200 BindingDB Entry DOI: 10.7270/Q2NS0VTJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50000129 (CHEMBL112763) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University College Dublin Curated by ChEMBL | Assay Description 25% inhibition of FGF-2 binding to heparin-albumin by ELISA | Bioorg Med Chem Lett 12: 3287-90 (2002) BindingDB Entry DOI: 10.7270/Q2ZP45G2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50454864 (CHEMBL4202957) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
CSIC and Universidad de Sevilla Curated by ChEMBL | Assay Description Inhibition of fluorescein labelled heparin-like hexasaccharide probe binding to recombinant human FGF-2 after 5 mins by fluorescence polarization ass... | Bioorg Med Chem 26: 1076-1085 (2018) Article DOI: 10.1016/j.bmc.2018.01.022 BindingDB Entry DOI: 10.7270/Q2H41V1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50454866 (CHEMBL4213376) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.71E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
CSIC and Universidad de Sevilla Curated by ChEMBL | Assay Description Inhibition of fluorescein labelled heparin-like hexasaccharide probe binding to recombinant human FGF-2 after 5 mins by fluorescence polarization ass... | Bioorg Med Chem 26: 1076-1085 (2018) Article DOI: 10.1016/j.bmc.2018.01.022 BindingDB Entry DOI: 10.7270/Q2H41V1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84561 (Linked sulfated tetracyclitol, 2) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84562 (Linked sulfated tetracyclitol, 3) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 248 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84563 (Linked sulfated tetracyclitol, 4) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 161 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84564 (Linked sulfated tetracyclitol, 5) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 148 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84565 (Linked sulfated tetracyclitol, 6) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 135 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84566 (Linked sulfated tetracyclitol, 7) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 90 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84567 (Linked sulfated tetracyclitol, 8) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 108 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84568 (Linked sulfated tetracyclitol, 9) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 194 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84569 (Linked sulfated tetracyclitol, 10) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 448 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84570 (Linked sulfated tetracyclitol, 11) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 332 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM84571 (Linked sulfated tetracyclitol, 12) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 85 | n/a | n/a | n/a | 7.4 | n/a |
Progen Industries Ltd. | Assay Description Human FGF-1 and FGF-2 were purchased from R&D Systems, Inc. and supplied as protein (ug) dissolved in bovine serum albumin (BSA, 50ug). Surface plas... | Chembiochem 6: 1882-90 (2005) Checked by Author Article DOI: 10.1002/cbic.200500089 BindingDB Entry DOI: 10.7270/Q22N50S0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50017346 (CHEMBL3288258) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.50E+7 | n/a | n/a | n/a | n/a | n/a |
Momenta Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity to human recombinant FGF2 by surface plasmon resonance assay | J Med Chem 57: 4511-20 (2014) Article DOI: 10.1021/jm4016069 BindingDB Entry DOI: 10.7270/Q2ZG6TSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor 2 (Homo sapiens (Human)) | BDBM50017347 (CHEMBL3288259) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Momenta Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity to human recombinant FGF2 by surface plasmon resonance assay | J Med Chem 57: 4511-20 (2014) Article DOI: 10.1021/jm4016069 BindingDB Entry DOI: 10.7270/Q2ZG6TSN | |||||||||||
More data for this Ligand-Target Pair |
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