Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122836 (CHEMBL102993 | [3-Carboxy-2-(3-tetradecyl-ureido)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MMDB PC cid PC sid UniChem Similars | Article PubMed | 360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver carnitine palmitoyltransferase I | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50033117 (CHEMBL114113 | [3-Carboxy-2-(hydroxy-tetradecyloxy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sandoz Research Institute Curated by ChEMBL | Assay Description In vitro inhibition of carnitine palmitoyltransferase I withrespect to palmitoyl CoA in rat | J Med Chem 38: 3448-50 (1995) BindingDB Entry DOI: 10.7270/Q2VQ31R1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50046145 (2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University Curated by ChEMBL | Assay Description Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat liver | J Med Chem 36: 237-42 (1993) BindingDB Entry DOI: 10.7270/Q2P849ZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50024430 ((R) (R) -2-Tetradecyl-oxirane-2-carboxylic acid-Co...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondria | J Med Chem 30: 1094-7 (1987) BindingDB Entry DOI: 10.7270/Q20P0Z1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50024434 ((+/-) 2-Tetradecyl-oxirane-2-carboxylic acid-Coenz...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondria | J Med Chem 30: 1094-7 (1987) BindingDB Entry DOI: 10.7270/Q20P0Z1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50024432 ((R)-(+)2-Tetradecyl-oxirane-2-carboxylic acid | CH...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondria | J Med Chem 30: 1094-7 (1987) BindingDB Entry DOI: 10.7270/Q20P0Z1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50024431 ((+/-)2-Tetradecyl-oxirane-2-carboxylic acid | 2-Te...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondria | J Med Chem 30: 1094-7 (1987) BindingDB Entry DOI: 10.7270/Q20P0Z1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50024429 ((R)-(+)2-Tetradecyl-oxirane-2-carboxylic acid meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondria | J Med Chem 30: 1094-7 (1987) BindingDB Entry DOI: 10.7270/Q20P0Z1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50024433 ((+/-) 2-Tetradecyl-oxirane-2-carboxylic acid methy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondria | J Med Chem 30: 1094-7 (1987) BindingDB Entry DOI: 10.7270/Q20P0Z1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50403029 (CHEMBL2216792) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT1A expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assay | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101604 (CHEMBL309568 | [3-Carboxy-2-(dodecane-1-sulfonylam...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101598 (CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101591 (CHEMBL308869 | R-[3-Carboxy-2-(undecane-1-sulfamoy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101591 (CHEMBL308869 | R-[3-Carboxy-2-(undecane-1-sulfamoy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122839 (CHEMBL106227 | [3-Carboxy-2-(3-tetradecyl-ureido)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50240113 (CHEMBL4081425) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
YachayTech University Curated by ChEMBL | Assay Description Inhibition of rat wild-type CPT1A expressed in yeast mitochondrial extracts using L-[methyl-3H]carnitine and palmitoyl-CoA as substrates preincubated... | Eur J Med Chem 131: 207-221 (2017) Article DOI: 10.1016/j.ejmech.2017.03.012 BindingDB Entry DOI: 10.7270/Q2TX3HHF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101594 (CHEMBL80493 | [3-Carboxy-2-(decane-1-sulfonylamino...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122834 (CHEMBL105314 | [3-Carboxy-2-(3-dodecyl-ureido)-pro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101589 (CHEMBL77174 | [3-Carboxy-2-(nonylaminosulphonyl-am...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122828 (CHEMBL106274 | [3-Carboxy-2-(3-undecyl-ureido)-pro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101600 (CHEMBL305897 | [3-Carboxy-2-(undecane-1-sulfamoyla...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101598 (CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101600 (CHEMBL305897 | [3-Carboxy-2-(undecane-1-sulfamoyla...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101604 (CHEMBL309568 | [3-Carboxy-2-(dodecane-1-sulfonylam...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122833 ((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50403046 (CHEMBL2216772) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT1A | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50240112 (CHEMBL4099442) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.57E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
YachayTech University Curated by ChEMBL | Assay Description Inhibition of rat wild-type CPT1A expressed in yeast mitochondrial extracts using L-[methyl-3H]carnitine and palmitoyl-CoA as substrates preincubated... | Eur J Med Chem 131: 207-221 (2017) Article DOI: 10.1016/j.ejmech.2017.03.012 BindingDB Entry DOI: 10.7270/Q2TX3HHF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101590 (CHEMBL78921 | [3-Carboxy-2-(3-nonyl-ureido)-propyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.95E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101593 ((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.23E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122827 (CHEMBL105330 | [3-Carboxy-2-(3-nonyl-ureido)-propy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.13E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50046145 (2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.85E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT1A using [3H]carnitine by radiometric assay | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50046145 (2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.85E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT1A using [3H]carnitine by radiometric assay | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122837 (CHEMBL319635 | [3-Carboxy-2-(3-heptyl-ureido)-prop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.36E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101597 ((3-Carboxy-2-tetradecyloxy-propyl)-trimethyl-ammon...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122836 (CHEMBL102993 | [3-Carboxy-2-(3-tetradecyl-ureido)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MMDB PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.88E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM61402 ((Z)-2-butenedioic acid;2-(2,2-dicyclohexylethyl)pi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of CPT1 in rat cardiac mitochondria using [3H]carnitine by radiometric method | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101607 (CHEMBL80353 | [3-Carboxy-2-(3-nonyl-thioureido)-pr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 1.22E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50284163 ((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article | n/a | n/a | 1.28E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II) | Bioorg Med Chem Lett 4: 883-886 (1994) Article DOI: 10.1016/S0960-894X(01)80256-0 BindingDB Entry DOI: 10.7270/Q2RX9C15 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM61402 ((Z)-2-butenedioic acid;2-(2,2-dicyclohexylethyl)pi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.48E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of CPT1 in rat liver mitochondria using [3H]carnitine by radiometric method | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101608 ((3-Carboxy-2-tetradecylamino-propyl)-trimethyl-amm...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM22984 ((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT1 in rat mitochondria | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101592 ((3-Carboxy-2-nonylcarbamoyloxy-propyl)-trimethyl-a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101596 (1-(3-Carboxy-2-tetradecyloxycarbonyloxy-propyl)-1-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101595 ((3-Carboxy-2-nonylcarbamoyloxy-propyl)-trimethyl-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122835 (CHEMBL105727 | [3-Carboxy-2-(3-nonyl-ureido)-propy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50122829 ((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondria | J Med Chem 46: 303-9 (2003) Article DOI: 10.1021/jm020979u BindingDB Entry DOI: 10.7270/Q2N015WM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101605 (1-(3-Phosphono-2-tetradecyloxycarbonyloxy-propyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101599 (CHEMBL77115 | Trimethyl-[2-tetradecyloxy-3-(2H-tet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101606 (CHEMBL80733 | Trimethyl-(2-nonylcarbamoyloxy-3-pho...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50101588 ((3-Carboxy-2-nonyloxycarbonyloxy-propyl)-trimethyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sigma Tau Pharmaceutical Industries S.p.A. Curated by ChEMBL | Assay Description Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligand | J Med Chem 44: 2383-6 (2001) BindingDB Entry DOI: 10.7270/Q2930SG7 | |||||||||||
More data for this Ligand-Target Pair |
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