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Compile Data Set for Download or QSAR

Found 1011 hits of affinity data for UniProtKB/TrEMBL: P52292   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75071
PNG
((6-ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 3,5-di...)
Show SMILES CCc1cc2c(COC(=O)c3c(C)noc3C)cc(=O)oc2cc1O
Show InChI InChI=1S/C18H17NO6/c1-4-11-5-13-12(6-16(21)24-15(13)7-14(11)20)8-23-18(22)17-9(2)19-25-10(17)3/h5-7,20H,4,8H2,1-3H3
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n/an/an/an/a 5.66E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75072
PNG
(2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-1-...)
Show SMILES CCOCCCNC(=O)NC(=O)CN1CCN(CC1)S(=O)(=O)c1ccc2OCCOc2c1
Show InChI InChI=1S/C20H30N4O7S/c1-2-29-11-3-6-21-20(26)22-19(25)15-23-7-9-24(10-8-23)32(27,28)16-4-5-17-18(14-16)31-13-12-30-17/h4-5,14H,2-3,6-13,15H2,1H3,(H2,21,22,25,26)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75073
PNG
(2-amino-5-keto-1-(4-methoxyphenyl)-2-pyrroline-3-c...)
Show SMILES COc1ccc(cc1)N1C(=O)CC(C#N)C1=N
Show InChI InChI=1S/C12H11N3O2/c1-17-10-4-2-9(3-5-10)15-11(16)6-8(7-13)12(15)14/h2-5,8,14H,6H2,1H3
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75074
PNG
((E)-3-(4-methylsulfanylphenyl)-2-[(5-phenyl-1,3,4-...)
Show SMILES CSc1ccc(\C=C(\Sc2nnc(o2)-c2ccccc2)C(O)=O)cc1
Show InChI InChI=1S/C18H14N2O3S2/c1-24-14-9-7-12(8-10-14)11-15(17(21)22)25-18-20-19-16(23-18)13-5-3-2-4-6-13/h2-11H,1H3,(H,21,22)/b15-11+
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n/an/an/an/a 4.10E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75075
PNG
(MLS001004634 | N'-(1,3-dimethyl-2,4-dioxo-6-pterid...)
Show SMILES Cn1c2ncc(NNC(=O)c3ccc(cc3)[N+]([O-])=O)nc2c(=O)n(C)c1=O
Show InChI InChI=1S/C15H13N7O5/c1-20-12-11(14(24)21(2)15(20)25)17-10(7-16-12)18-19-13(23)8-3-5-9(6-4-8)22(26)27/h3-7H,1-2H3,(H,17,18)(H,19,23)
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n/an/an/an/a 5.42E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM36913
PNG
(2-[(2,5-dimethyl-1-pyridin-2-yl-pyrrol-3-yl)methyl...)
Show SMILES Cc1cc(C=c2sc3nc4ccccc4n3c2=O)c(C)n1-c1ccccn1
Show InChI InChI=1S/C21H16N4OS/c1-13-11-15(14(2)24(13)19-9-5-6-10-22-19)12-18-20(26)25-17-8-4-3-7-16(17)23-21(25)27-18/h3-12H,1-2H3
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n/an/an/an/a 1.83E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75076
PNG
(2-(3-pyridyl)-N-(2-thiazolin-2-yl)cinchoninamide;h...)
Show SMILES O=C(NC1=NCCS1)c1cc(nc2ccccc12)-c1cccnc1 |t:3|
Show InChI InChI=1S/C18H14N4OS/c23-17(22-18-20-8-9-24-18)14-10-16(12-4-3-7-19-11-12)21-15-6-2-1-5-13(14)15/h1-7,10-11H,8-9H2,(H,20,22,23)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75077
PNG
(5-cyano-4-(2-furanyl)-N,2-dimethyl-6-sulfanylidene...)
Show SMILES CNC(=O)c1c(C)[nH]c(=S)c(C#N)c1-c1ccco1
Show InChI InChI=1S/C13H11N3O2S/c1-7-10(12(17)15-2)11(9-4-3-5-18-9)8(6-14)13(19)16-7/h3-5H,1-2H3,(H,15,17)(H,16,19)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75078
PNG
(10-[3-(diisoamylamino)-2-hydroxy-propyl]acridin-9-...)
Show SMILES CC(C)CCN(CCC(C)C)CC(O)Cn1c2ccccc2c(=O)c2ccccc12
Show InChI InChI=1S/C26H36N2O2/c1-19(2)13-15-27(16-14-20(3)4)17-21(29)18-28-24-11-7-5-9-22(24)26(30)23-10-6-8-12-25(23)28/h5-12,19-21,29H,13-18H2,1-4H3
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n/an/an/an/a 3.74E+3n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM50593
PNG
(4-Methyl-benzoic acid N'-acridin-9-yl-hydrazid...)
Show SMILES Cc1ccc(cc1)C(=O)NNc1c2ccccc2nc2ccccc12
Show InChI InChI=1S/C21H17N3O/c1-14-10-12-15(13-11-14)21(25)24-23-20-16-6-2-4-8-18(16)22-19-9-5-3-7-17(19)20/h2-13H,1H3,(H,22,23)(H,24,25)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM52775
PNG
(3-Imino-1,5,7-trimethyl-2,6-dioxa-bicyclo[2.2.2]oc...)
Show SMILES CC1OC2(C)OC(=N)C1(C#N)C(C#N)(C#N)C2C |TLB:7:6:16.11:2.1,0:1:16.11:5.6,THB:17:16:2.1:5.6|
Show InChI InChI=1S/C12H12N4O2/c1-7-10(3)17-8(2)12(6-15,9(16)18-10)11(7,4-13)5-14/h7-8,16H,1-3H3
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n/an/an/an/a 7.74E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM63780
PNG
(3-[4-(trifluoromethyl)phenyl]-N-[[2-(trifluorometh...)
Show SMILES FC(F)(F)c1ccc(cc1)C1=NOC(C1)C(=O)NCc1ccccc1C(F)(F)F |t:11|
Show InChI InChI=1S/C19H14F6N2O2/c20-18(21,22)13-7-5-11(6-8-13)15-9-16(29-27-15)17(28)26-10-12-3-1-2-4-14(12)19(23,24)25/h1-8,16H,9-10H2,(H,26,28)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75079
PNG
((5E)-5-[(1-azepanylamino)methylidene]-1-(1-naphtha...)
Show SMILES Oc1c(C=NN2CCCCCC2)c(=O)[nH]c(=O)n1-c1cccc2ccccc12 |w:4.4,(7.72,1.65,;9.05,.88,;9.05,-.66,;7.72,-1.43,;7.72,-2.97,;6.39,-3.74,;5.11,-2.87,;3.64,-3.33,;3.08,-4.76,;3.85,-6.09,;5.37,-6.32,;6.5,-5.28,;10.39,-1.43,;10.39,-2.97,;11.72,-.66,;11.72,.88,;13.06,1.65,;10.39,1.65,;10.39,3.19,;9.05,3.96,;9.05,5.5,;10.39,6.27,;11.72,5.5,;13.1,6.32,;14.49,5.53,;14.49,3.93,;13.1,3.14,;11.72,3.96,)|
Show InChI InChI=1S/C21H22N4O3/c26-19-17(14-22-24-12-5-1-2-6-13-24)20(27)25(21(28)23-19)18-11-7-9-15-8-3-4-10-16(15)18/h3-4,7-11,14,27H,1-2,5-6,12-13H2,(H,23,26,28)/b22-14+
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM58045
PNG
(2-Amino-1-(3-methoxy-propyl)-1H-pyrrolo[2,3-b]quin...)
Show SMILES COCCCn1c(N)c(C(=O)Nc2ccccc2)c2nc3ccccc3nc12
Show InChI InChI=1S/C21H21N5O2/c1-28-13-7-12-26-19(22)17(21(27)23-14-8-3-2-4-9-14)18-20(26)25-16-11-6-5-10-15(16)24-18/h2-6,8-11H,7,12-13,22H2,1H3,(H,23,27)
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n/an/an/an/a 2.53E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75080
PNG
((Z)-4-(4-cyanophenyl)-2-keto-3-(2-quinolyl)but-3-e...)
Show SMILES OC(=O)C(=O)C(=C/c1ccc(cc1)C#N)\c1ccc2ccccc2n1
Show InChI InChI=1S/C20H12N2O3/c21-12-14-7-5-13(6-8-14)11-16(19(23)20(24)25)18-10-9-15-3-1-2-4-17(15)22-18/h1-11H,(H,24,25)/b16-11-
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n/an/an/an/a 1.25E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75081
PNG
(2-[2-(3-ethanoylphenoxy)ethanoyl-methyl-amino]-N-(...)
Show SMILES CN(CC(=O)Nc1ccc(F)cc1)C(=O)COc1cccc(c1)C(C)=O
Show InChI InChI=1S/C19H19FN2O4/c1-13(23)14-4-3-5-17(10-14)26-12-19(25)22(2)11-18(24)21-16-8-6-15(20)7-9-16/h3-10H,11-12H2,1-2H3,(H,21,24)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75082
PNG
(2-[[(E)-(6-keto-4-methyl-cyclohexa-2,4-dien-1-ylid...)
Show SMILES CCOC(=O)c1c2CCN(C)Cc2sc1N=Cc1ccc(C)cc1O |w:15.16|
Show InChI InChI=1S/C19H22N2O3S/c1-4-24-19(23)17-14-7-8-21(3)11-16(14)25-18(17)20-10-13-6-5-12(2)9-15(13)22/h5-6,9-10,22H,4,7-8,11H2,1-3H3
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n/an/an/an/a>2.60E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75083
PNG
(3-cyclohexyl-2-diazanyl-7-(phenylmethyl)-6,8-dihyd...)
Show SMILES NNc1nc2sc3CN(Cc4ccccc4)CCc3c2c(=O)n1C1CCCCC1
Show InChI InChI=1S/C22H27N5OS/c23-25-22-24-20-19(21(28)27(22)16-9-5-2-6-10-16)17-11-12-26(14-18(17)29-20)13-15-7-3-1-4-8-15/h1,3-4,7-8,16H,2,5-6,9-14,23H2,(H,24,25)
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n/an/an/an/a 918n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75084
PNG
(MLS001012124 | SMR000425279 | [5-(4-Bromo-phenyl)-...)
Show SMILES CC1=NN(C(=O)c2ccccc2)C(O)(C1)c1ccc(Br)cc1 |t:1|
Show InChI InChI=1S/C17H15BrN2O2/c1-12-11-17(22,14-7-9-15(18)10-8-14)20(19-12)16(21)13-5-3-2-4-6-13/h2-10,22H,11H2,1H3
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75085
PNG
((E)-2-Cyano-3-(9-methyl-4-oxo-2-phenoxy-4H-pyrido[...)
Show SMILES Cc1cccn2c1nc(Oc1ccccc1)c(\C=C(/C#N)C(N)=O)c2=O
Show InChI InChI=1S/C19H14N4O3/c1-12-6-5-9-23-17(12)22-18(26-14-7-3-2-4-8-14)15(19(23)25)10-13(11-20)16(21)24/h2-10H,1H3,(H2,21,24)/b13-10+
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n/an/an/an/a 1.58E+3n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM60208
PNG
(2-[2-(1-Allyl-1H-pyridin-4-ylidene)-ethylidene]-ma...)
Show SMILES [#6]=[#6]-[#6]-[#7]-1-[#6]=[#6]\[#6](=[#6]\[#6]=[#6](\C#N)C#N)-[#6]=[#6]-1 |c:4,14|
Show InChI InChI=1S/C13H11N3/c1-2-7-16-8-5-12(6-9-16)3-4-13(10-14)11-15/h2-6,8-9H,1,7H2
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n/an/an/an/a 1.67E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75086
PNG
(1-(1-Amino-5-methyl-6,7,8,9-tetrahydro-thieno[2,3-...)
Show SMILES CC(=O)c1sc2nc(C)c3CCCCc3c2c1N
Show InChI InChI=1S/C14H16N2OS/c1-7-9-5-3-4-6-10(9)11-12(15)13(8(2)17)18-14(11)16-7/h3-6,15H2,1-2H3
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n/an/an/an/a 1.44E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75087
PNG
(2-(2-Fluoro-phenyl)-5,6-dimethyl-2,3-dihydro-1H-th...)
Show SMILES Cc1sc2NC(NC(=O)c2c1C)c1ccccc1F
Show InChI InChI=1S/C14H13FN2OS/c1-7-8(2)19-14-11(7)13(18)16-12(17-14)9-5-3-4-6-10(9)15/h3-6,12,17H,1-2H3,(H,16,18)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75088
PNG
(MLS000333714 | Morpholin-4-yl-acetic acid N'-a...)
Show SMILES O=C(CN1CCOCC1)NNc1c2ccccc2nc2ccccc12
Show InChI InChI=1S/C19H20N4O2/c24-18(13-23-9-11-25-12-10-23)21-22-19-14-5-1-3-7-16(14)20-17-8-4-2-6-15(17)19/h1-8H,9-13H2,(H,20,22)(H,21,24)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75089
PNG
(MLS000780334 | N-[4-[[(E)-N'-(4,6-dimethylpyrimidi...)
Show SMILES CCC(=O)Nc1ccc(cc1)N=C(N)Nc1nc(C)cc(C)n1 |w:11.11|
Show InChI InChI=1S/C16H20N6O/c1-4-14(23)20-12-5-7-13(8-6-12)21-15(17)22-16-18-10(2)9-11(3)19-16/h5-9H,4H2,1-3H3,(H,20,23)(H3,17,18,19,21,22)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75090
PNG
(4-Hydroxy-butyric acid N'-acridin-9-yl-hydrazi...)
Show SMILES OCCCC(=O)NNc1c2ccccc2nc2ccccc12
Show InChI InChI=1S/C17H17N3O2/c21-11-5-10-16(22)19-20-17-12-6-1-3-8-14(12)18-15-9-4-2-7-13(15)17/h1-4,6-9,21H,5,10-11H2,(H,18,20)(H,19,22)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75091
PNG
((5E)-5-[(1-azepanylamino)methylidene]-1-(3,4-dimet...)
Show SMILES Cc1ccc(cc1C)-n1c(O)c(C=NN2CCCCCC2)c(=O)[nH]c1=O |w:13.14|
Show InChI InChI=1S/C19H24N4O3/c1-13-7-8-15(11-14(13)2)23-18(25)16(17(24)21-19(23)26)12-20-22-9-5-3-4-6-10-22/h7-8,11-12,25H,3-6,9-10H2,1-2H3,(H,21,24,26)/b20-12+
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75092
PNG
(2-Amino-benzoic acid N'-acridin-9-yl-hydrazide...)
Show SMILES Nc1ccccc1C(=O)NNc1c2ccccc2nc2ccccc12
Show InChI InChI=1S/C20H16N4O/c21-16-10-4-1-7-13(16)20(25)24-23-19-14-8-2-5-11-17(14)22-18-12-6-3-9-15(18)19/h1-12H,21H2,(H,22,23)(H,24,25)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75093
PNG
(Adamantane-1-carboxylic acid N'-acridin-9-yl-h...)
Show SMILES [H]C12CC3([H])CC([H])(C1)CC(C2)(C3)C(=O)NNc1c2ccccc2nc2ccccc12 |TLB:5:3:11:6.9.8,8:1:12:6.9.5,8:6:12:1.11.2,THB:5:6:11:3.12.2,2:1:9:3.12.5|
Show InChI InChI=1S/C24H25N3O/c28-23(24-12-15-9-16(13-24)11-17(10-15)14-24)27-26-22-18-5-1-3-7-20(18)25-21-8-4-2-6-19(21)22/h1-8,15-17H,9-14H2,(H,25,26)(H,27,28)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75094
PNG
((E)-2-Cyano-N-cyclohexyl-3-(5-morpholin-4-yl-furan...)
Show SMILES O=C(NC1CCCCC1)C(=C\c1ccc(o1)N1CCOCC1)\C#N
Show InChI InChI=1S/C18H23N3O3/c19-13-14(18(22)20-15-4-2-1-3-5-15)12-16-6-7-17(24-16)21-8-10-23-11-9-21/h6-7,12,15H,1-5,8-11H2,(H,20,22)/b14-12+
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n/an/an/an/a 3.85E+3n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75095
PNG
((5Z)-3-(3-methylphenyl)-5-(3-pyridinylmethylidene)...)
Show SMILES Cc1cccc(c1)N1C(=S)S\C(=C/c2cccnc2)C1=O
Show InChI InChI=1S/C16H12N2OS2/c1-11-4-2-6-13(8-11)18-15(19)14(21-16(18)20)9-12-5-3-7-17-10-12/h2-10H,1H3/b14-9-
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75096
PNG
((E)-2-Cyano-3-(5-dimethylamino-furan-2-yl)-N-isopr...)
Show SMILES CC(C)NC(=O)C(=C\c1ccc(o1)N(C)C)\C#N
Show InChI InChI=1S/C13H17N3O2/c1-9(2)15-13(17)10(8-14)7-11-5-6-12(18-11)16(3)4/h5-7,9H,1-4H3,(H,15,17)/b10-7+
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n/an/an/an/a 6.38E+3n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75097
PNG
((E)-2-Cyano-3-[2-(4-methoxy-phenoxy)-9-methyl-4-ox...)
Show SMILES COc1ccc(Oc2nc3c(C)cccn3c(=O)c2\C=C(/C#N)C(N)=O)cc1
Show InChI InChI=1S/C20H16N4O4/c1-12-4-3-9-24-18(12)23-19(28-15-7-5-14(27-2)6-8-15)16(20(24)26)10-13(11-21)17(22)25/h3-10H,1-2H3,(H2,22,25)/b13-10+
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n/an/an/an/a 6.00E+3n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75098
PNG
(MLS000332669 | N-(1-Ethyl-8-methyl-1H-pyrazolo[3,4...)
Show SMILES CCn1nc(NC(=O)Cc2ccc(OC)cc2)c2cc3cccc(C)c3nc12
Show InChI InChI=1S/C22H22N4O2/c1-4-26-22-18(13-16-7-5-6-14(2)20(16)24-22)21(25-26)23-19(27)12-15-8-10-17(28-3)11-9-15/h5-11,13H,4,12H2,1-3H3,(H,23,25,27)
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n/an/an/an/a 5.90E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75099
PNG
(MLS000737612 | N-(4-ethoxyphenyl)-9-acridinamine |...)
Show SMILES CCOc1ccc(Nc2c3ccccc3nc3ccccc23)cc1
Show InChI InChI=1S/C21H18N2O/c1-2-24-16-13-11-15(12-14-16)22-21-17-7-3-5-9-19(17)23-20-10-6-4-8-18(20)21/h3-14H,2H2,1H3,(H,22,23)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75100
PNG
(2-Amino-1-(3-morpholin-4-yl-propyl)-1H-pyrrolo[2,3...)
Show SMILES Nc1c(C(=O)Nc2ccccc2)c2nc3ccccc3nc2n1CCCN1CCOCC1
Show InChI InChI=1S/C24H26N6O2/c25-22-20(24(31)26-17-7-2-1-3-8-17)21-23(28-19-10-5-4-9-18(19)27-21)30(22)12-6-11-29-13-15-32-16-14-29/h1-5,7-10H,6,11-16,25H2,(H,26,31)
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n/an/an/an/a 2.96E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75101
PNG
((2Z)-2-(2-furanylmethylidene)-6-methoxy-3-benzofur...)
Show SMILES COc1ccc2C(=O)\C(Oc2c1)=C\c1ccco1
Show InChI InChI=1S/C14H10O4/c1-16-9-4-5-11-12(7-9)18-13(14(11)15)8-10-3-2-6-17-10/h2-8H,1H3/b13-8-
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n/an/an/an/a 1.88E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM73775
PNG
((E)-2-Cyano-3-(1-methyl-5-p-tolyl-1H-pyrrol-2-yl)-...)
Show SMILES Cc1ccc(cc1)-c1ccc(\C=C(/C#N)C(N)=S)n1C
Show InChI InChI=1S/C16H15N3S/c1-11-3-5-12(6-4-11)15-8-7-14(19(15)2)9-13(10-17)16(18)20/h3-9H,1-2H3,(H2,18,20)/b13-9+
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75102
PNG
(Acridin-9-yl-[2-(3,4-dimethoxy-phenyl)-ethyl]-amin...)
Show SMILES COc1ccc(CCNc2c3ccccc3nc3ccccc23)cc1OC
Show InChI InChI=1S/C23H22N2O2/c1-26-21-12-11-16(15-22(21)27-2)13-14-24-23-17-7-3-5-9-19(17)25-20-10-6-4-8-18(20)23/h3-12,15H,13-14H2,1-2H3,(H,24,25)
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n/an/an/an/a 1.44E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM52844
PNG
(4-[(5,6-dioxo-3-pyridinyl)hydrazo]benzenesulfonami...)
Show SMILES NS(=O)(=O)c1ccc(cc1)N=Nc1c[nH]c(=O)c(O)c1 |w:10.10|
Show InChI InChI=1S/C11H10N4O4S/c12-20(18,19)9-3-1-7(2-4-9)14-15-8-5-10(16)11(17)13-6-8/h1-6,16H,(H,13,17)(H2,12,18,19)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75103
PNG
(3-(1,3-benzothiazol-2-yl)-7-hydroxy-8-[(2-methyl-1...)
Show SMILES CC1CCCCN1Cc1c(O)ccc2c1occ(-c1nc3ccccc3s1)c2=O
Show InChI InChI=1S/C23H22N2O3S/c1-14-6-4-5-11-25(14)12-16-19(26)10-9-15-21(27)17(13-28-22(15)16)23-24-18-7-2-3-8-20(18)29-23/h2-3,7-10,13-14,26H,4-6,11-12H2,1H3
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n/an/an/an/a<380n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM54113
PNG
(6-Chloro-8-diethylaminomethyl-7-hydroxy-4-propyl-c...)
Show SMILES CCCc1cc(=O)oc2c(CN(CC)CC)c(O)c(Cl)cc12
Show InChI InChI=1S/C17H22ClNO3/c1-4-7-11-8-15(20)22-17-12(11)9-14(18)16(21)13(17)10-19(5-2)6-3/h8-9,21H,4-7,10H2,1-3H3
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n/an/an/an/a 5.67E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM50194826
PNG
(2-amino-4-(4-fluorophenyl)-6,7-dihydro-5H-cyclopen...)
Show SMILES Nc1nc2CCCc2c(-c2ccc(F)cc2)c1C#N
Show InChI InChI=1S/C15H12FN3/c16-10-6-4-9(5-7-10)14-11-2-1-3-13(11)19-15(18)12(14)8-17/h4-7H,1-3H2,(H2,18,19)
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n/an/an/an/a 9.91E+3n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75104
PNG
(7-Methyl-2-[4-(3,4,5-trimethoxy-benzoyl)-[1,4]diaz...)
Show SMILES COc1cc(cc(OC)c1OC)C(=O)N1CCCN(CC1)c1nc2cc(C)ccc2cc1C#N
Show InChI InChI=1S/C26H28N4O4/c1-17-6-7-18-13-20(16-27)25(28-21(18)12-17)29-8-5-9-30(11-10-29)26(31)19-14-22(32-2)24(34-4)23(15-19)33-3/h6-7,12-15H,5,8-11H2,1-4H3
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n/an/an/an/a 1.54E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75105
PNG
(4-(3-bromo-4,5-dimethoxy-phenyl)-1-(2-methoxyethyl...)
Show SMILES COCCN1C=C(C(C(=C1)C(=O)OC)c1cc(Br)c(OC)c(OC)c1)C(=O)OC |c:5,8|
Show InChI InChI=1S/C20H24BrNO7/c1-25-7-6-22-10-13(19(23)28-4)17(14(11-22)20(24)29-5)12-8-15(21)18(27-3)16(9-12)26-2/h8-11,17H,6-7H2,1-5H3
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n/an/an/an/a 3.05E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75106
PNG
(3-[(2Z)-2-(4-keto-2-thioxo-thiazolidin-5-ylidene)-...)
Show SMILES OS(=O)(=O)CCCN1C(Sc2ccccc12)=C1SC(S)=NC1=O |w:8.8,c:21|
Show InChI InChI=1S/C13H12N2O4S4/c16-11-10(22-13(20)14-11)12-15(6-3-7-23(17,18)19)8-4-1-2-5-9(8)21-12/h1-2,4-5H,3,6-7H2,(H,14,16,20)(H,17,18,19)
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n/an/an/an/a 1.49E+4n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75107
PNG
(2-(cyclohexylamino)-N-[3-(dimethylsulfamoyl)phenyl...)
Show SMILES CN(C)S(=O)(=O)c1cccc(NC(=O)CNC2CCCCC2)c1
Show InChI InChI=1S/C16H25N3O3S/c1-19(2)23(21,22)15-10-6-9-14(11-15)18-16(20)12-17-13-7-4-3-5-8-13/h6,9-11,13,17H,3-5,7-8,12H2,1-2H3,(H,18,20)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75108
PNG
(MLS001005988 | N-(9-ethyl-3-carbazolyl)-2-(methyla...)
Show SMILES CCn1c2ccccc2c2cc(NC(=O)CNC)ccc12
Show InChI InChI=1S/C17H19N3O/c1-3-20-15-7-5-4-6-13(15)14-10-12(8-9-16(14)20)19-17(21)11-18-2/h4-10,18H,3,11H2,1-2H3,(H,19,21)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75109
PNG
(2-(2-bromanyl-4-fluoranyl-phenoxy)ethanoic acid | ...)
Show SMILES OC(=O)COc1ccc(F)cc1Br
Show InChI InChI=1S/C8H6BrFO3/c9-6-3-5(10)1-2-7(6)13-4-8(11)12/h1-3H,4H2,(H,11,12)
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MCE
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM50693
PNG
((5Z)-2-(4-fluoroanilino)-5-(1H-indol-3-ylmethylene...)
Show SMILES Fc1ccc(NC2=NC(=O)C(S2)=Cc2c[nH]c3ccccc23)cc1 |w:12.13,t:6|
Show InChI InChI=1S/C18H12FN3OS/c19-12-5-7-13(8-6-12)21-18-22-17(23)16(24-18)9-11-10-20-15-4-2-1-3-14(11)15/h1-10,20H,(H,21,22,23)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair
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