Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169013 (CHEMBL3805703) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Competitive inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) assessed as formation of G6P by continuou... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169042 (CHEMBL3806103) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169037 (CHEMBL3805205) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169031 (CHEMBL3805905) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169041 (CHEMBL3805653) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169038 (CHEMBL3804841) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169039 (CHEMBL3806132) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169043 (CHEMBL3806095) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169034 (CHEMBL3805734) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169032 (CHEMBL3805398) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169026 (CHEMBL3805148) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169046 (CHEMBL3805459) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169040 (CHEMBL3804874) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169033 (CHEMBL3806069) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169031 (CHEMBL3805905) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of HK2 in human UM-UC-3 cells using 2FDG as substrate assessed as suppression of G6P production preincubated for 30 mins followed by subst... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50103565 (CHEMBL3335788) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >316 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Pisa Curated by ChEMBL | Assay Description Inhibition of hexokinase 2 (unknown origin) | Bioorg Med Chem Lett 24: 4915-25 (2014) Article DOI: 10.1016/j.bmcl.2014.09.041 BindingDB Entry DOI: 10.7270/Q25Q4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169028 (CHEMBL3805598) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169041 (CHEMBL3805653) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 470 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of HK2 in human UM-UC-3 cells using 2FDG as substrate assessed as suppression of G6P production preincubated for 30 mins followed by subst... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169046 (CHEMBL3805459) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 520 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of HK2 in human UM-UC-3 cells using 2FDG as substrate assessed as suppression of G6P production preincubated for 30 mins followed by subst... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169036 (CHEMBL3806028) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 630 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169023 (CHEMBL3805753) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 790 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169017 (CHEMBL3804930) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 790 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169025 (CHEMBL3806250) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169019 (CHEMBL3805765) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169015 (CHEMBL3805460) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512392 (CHEMBL4474580) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM49122 (2-amino-3-hydroxy-N'-(2,3,4-trihydroxybenzyl)propi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shandong University at Weihai Curated by ChEMBL | Assay Description Inhibition of HK2 (unknown origin) using glucose-6-phosphate dehydrogenase as substrate preincubated for 10 mins followed by substrate addition | J Nat Prod 82: 1114-1119 (2019) Article DOI: 10.1021/acs.jnatprod.8b00821 BindingDB Entry DOI: 10.7270/Q20G3PD7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169013 (CHEMBL3805703) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512405 (CHEMBL4466819) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.36E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50505250 (CHEMBL4447523) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shandong University at Weihai Curated by ChEMBL | Assay Description Inhibition of HK2 (unknown origin) using glucose-6-phosphate dehydrogenase as substrate preincubated for 10 mins followed by substrate addition | J Nat Prod 82: 1114-1119 (2019) Article DOI: 10.1021/acs.jnatprod.8b00821 BindingDB Entry DOI: 10.7270/Q20G3PD7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169018 (CHEMBL3804924) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50169014 (CHEMBL3806183) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a... | ACS Med Chem Lett 7: 217-22 (2016) Article DOI: 10.1021/acsmedchemlett.5b00214 BindingDB Entry DOI: 10.7270/Q2PR7XWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512404 (CHEMBL4439269) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.61E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50505249 (CHEMBL4435293) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.12E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shandong University at Weihai Curated by ChEMBL | Assay Description Inhibition of HK2 (unknown origin) using glucose-6-phosphate dehydrogenase as substrate preincubated for 10 mins followed by substrate addition | J Nat Prod 82: 1114-1119 (2019) Article DOI: 10.1021/acs.jnatprod.8b00821 BindingDB Entry DOI: 10.7270/Q20G3PD7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50505248 (CHEMBL4557294) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.46E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shandong University at Weihai Curated by ChEMBL | Assay Description Inhibition of HK2 (unknown origin) using glucose-6-phosphate dehydrogenase as substrate preincubated for 10 mins followed by substrate addition | J Nat Prod 82: 1114-1119 (2019) Article DOI: 10.1021/acs.jnatprod.8b00821 BindingDB Entry DOI: 10.7270/Q20G3PD7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512389 (CHEMBL4441499) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512390 (CHEMBL4559740) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512391 (CHEMBL4440088) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50084419 (Andrographolide | CHEBI:65408) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512393 (CHEMBL4435724) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512394 (CHEMBL4458194) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512396 (CHEMBL4473377) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512397 (CHEMBL4573718) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512398 (CHEMBL4457024) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512399 (CHEMBL4440743) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512400 (CHEMBL4448145) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512401 (CHEMBL4592431) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512402 (CHEMBL4580347) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512403 (CHEMBL4565147) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-2 (Homo sapiens (Human)) | BDBM50512388 (CHEMBL4476790) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shenyang Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate... | Eur J Med Chem 173: 282-293 (2019) Article DOI: 10.1016/j.ejmech.2019.04.022 BindingDB Entry DOI: 10.7270/Q2Z322ZG | |||||||||||
More data for this Ligand-Target Pair |
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