Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Growth factor receptor-bound protein 10 (Homo sapiens (Human)) | BDBM50124406 (CHEMBL3623450) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 4.20E+5 | n/a | n/a | n/a | n/a | n/a |
The University of Sydney Curated by ChEMBL | Assay Description Binding affinity to GST-tagged Grb10-SH2 domain (471 to 594 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 m... | J Med Chem 58: 7707-18 (2015) Article DOI: 10.1021/acs.jmedchem.5b00609 BindingDB Entry DOI: 10.7270/Q23X88GG | |||||||||||
More data for this Ligand-Target Pair |