Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574750 (CHEMBL4850758) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 293 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Mixed inhibition of human KDM4D expressed in Escherichia coli BL21(DE3) using H3(1-21)K9me3 peptide and varying concentrations of 2-OG as substrate p... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50598656 (CHEMBL5206330) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c00680 BindingDB Entry DOI: 10.7270/Q2W95F76 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574750 (CHEMBL4850758) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM293660 (3-({[(1S)-6-[methyl(phenyl)amino]-1,2,3,4-tetrahyd...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c00680 BindingDB Entry DOI: 10.7270/Q2W95F76 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574748 (CHEMBL4875100) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574753 (CHEMBL4866032) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50153322 (CHEMBL3775612) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of human KDM4D (11 to 341 residues) using H3K9Me3 peptide as substrate assessed as demethylation of substrate by Rapidfire mass spectromet... | J Med Chem 59: 1357-69 (2016) Article DOI: 10.1021/acs.jmedchem.5b01537 BindingDB Entry DOI: 10.7270/Q2542QFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50153318 (CHEMBL3775237) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c00680 BindingDB Entry DOI: 10.7270/Q2W95F76 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574755 (CHEMBL4852549) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 87 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50153318 (CHEMBL3775237) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of human KDM4D (11 to 341 residues) using H3K9Me3 peptide as substrate assessed as demethylation of substrate by Rapidfire mass spectromet... | J Med Chem 59: 1357-69 (2016) Article DOI: 10.1021/acs.jmedchem.5b01537 BindingDB Entry DOI: 10.7270/Q2542QFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50153319 (CHEMBL3775889) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of human KDM4D (11 to 341 residues) using H3K9Me3 peptide as substrate assessed as demethylation of substrate by Rapidfire mass spectromet... | J Med Chem 59: 1357-69 (2016) Article DOI: 10.1021/acs.jmedchem.5b01537 BindingDB Entry DOI: 10.7270/Q2542QFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574749 (CHEMBL4865890) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM293660 (3-({[(1S)-6-[methyl(phenyl)amino]-1,2,3,4-tetrahyd...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 104 | n/a | n/a | n/a | n/a | n/a | n/a |
Celgene Quanticel Research Curated by ChEMBL | Assay Description Inhibition of KDM4D (unknown origin) using biotinylated H3K9me3 peptide and alpha-ketoglutarate as substrate pretreated for 1 hr followed by substrat... | ACS Med Chem Lett 8: 869-874 (2017) Article DOI: 10.1021/acsmedchemlett.7b00220 BindingDB Entry DOI: 10.7270/Q2HH6NPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574756 (CHEMBL4849386) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 109 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM191600 (2-(5-((4-chloro-2-methylbenzyl)oxy)-1Hpyrazol-1-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Celgene Corporation Curated by ChEMBL | Assay Description Inhibition of KDM4D (unknown origin) | Bioorg Med Chem Lett 28: 1490-1494 (2018) Article DOI: 10.1016/j.bmcl.2018.03.083 BindingDB Entry DOI: 10.7270/Q26Q20W4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574738 (CHEMBL4863496) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 111 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574739 (CHEMBL4853213) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 117 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574757 (CHEMBL4870370) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574709 (CHEMBL4851604) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 135 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574740 (CHEMBL4848874) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 141 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574752 (CHEMBL4870256) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 145 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574710 (CHEMBL4865527) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 155 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574758 (CHEMBL4867448) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 165 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574721 (CHEMBL4852779) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574727 (CHEMBL4853385) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 171 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574736 (CHEMBL4867797) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 173 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574759 (CHEMBL4864457) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 184 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574718 (CHEMBL4869955) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 187 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574726 (CHEMBL4879231) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 188 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574737 (CHEMBL4847665) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 192 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574723 (CHEMBL4857387) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 193 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50396018 (CHEMBL1230640) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01204 BindingDB Entry DOI: 10.7270/Q2BR8X83 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50153339 (CHEMBL3775431) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of human KDM4D (11 to 341 residues) using H3K9Me3 peptide as substrate assessed as demethylation of substrate by Rapidfire mass spectromet... | J Med Chem 59: 1357-69 (2016) Article DOI: 10.1021/acs.jmedchem.5b01537 BindingDB Entry DOI: 10.7270/Q2542QFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574730 (CHEMBL4866118) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574734 (CHEMBL4865163) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 212 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574712 (CHEMBL4866179) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574751 (CHEMBL4853701) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574760 (CHEMBL4850795) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 223 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50153341 (CHEMBL3774845) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 251 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of human KDM4D (11 to 341 residues) using H3K9Me3 peptide as substrate assessed as demethylation of substrate by Rapidfire mass spectromet... | J Med Chem 59: 1357-69 (2016) Article DOI: 10.1021/acs.jmedchem.5b01537 BindingDB Entry DOI: 10.7270/Q2542QFT | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574761 (CHEMBL4871665) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 285 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50498665 (CHEMBL1982368) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of KDM4D (unknown origin) | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50498665 (CHEMBL1982368) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c00680 BindingDB Entry DOI: 10.7270/Q2W95F76 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50149925 (CHEMBL3770740) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of KDM4D (unknown origin) by RFMS assay | J Med Chem 59: 1370-87 (2016) Article DOI: 10.1021/acs.jmedchem.5b01538 BindingDB Entry DOI: 10.7270/Q26D5VV2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574742 (CHEMBL4851379) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574722 (CHEMBL4876010) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 342 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574716 (CHEMBL4857330) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 351 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574743 (CHEMBL4878349) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 368 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50574741 (CHEMBL4870942) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 382 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113662 BindingDB Entry DOI: 10.7270/Q24T6P5X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM195612 (GSK467) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 398 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of KDM4D (unknown origin) by RFMS assay | J Med Chem 59: 1370-87 (2016) Article DOI: 10.1021/acs.jmedchem.5b01538 BindingDB Entry DOI: 10.7270/Q26D5VV2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 4D (Homo sapiens (Human)) | BDBM50149917 (CHEMBL3771198) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 398 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of KDM4D (unknown origin) by RFMS assay | J Med Chem 59: 1370-87 (2016) Article DOI: 10.1021/acs.jmedchem.5b01538 BindingDB Entry DOI: 10.7270/Q26D5VV2 | |||||||||||
More data for this Ligand-Target Pair |
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