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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
Compound
FDA Drugs
Important Compounds
Chemical Structure
Name
SMILES
Number of Data
/
Targets
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3D Structure Series
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Citation
Author
Journal/Citation
Institution
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Special Data Sets
D3R
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Prot-Lig Validation Sets
Other Databases
PDB
85%
100%
Seq ID
UniProtKB/Swiss-Prot
UniProtKB/TrEMBL
PubMed
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All Compounds & Data
Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Deposition
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Sent Comments
UniProtKB/Swiss_Prot/TrEMBL Accession Numbers in Gamma-secretase
A4D1B5
A4D1B6
A8K8D4
B1AP21
B2R5L9
B2R5V1
B4DII8
D3DSD1
D3DSD2
D3DSD3
P05067
P09000
P49768
P49810
P78438
Q13764
Q13778
Q13793
Q16011
Q16014
Q16019
Q16020
Q3MJC0
Q6GSC0
Q8ND73
Q8WW43
Q8WZ99
Q92542
Q96BI3
Q96P32
Q9BT38
Q9NZ42
Q9UC33
Q9UCA9
Q9UCB6
Q9UCC8
Q9UCD1
Q9UMH3
Q9UQ58
Q9Y4L9