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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
Compound
FDA Drugs
Important Compounds
Chemical Structure
Name
SMILES
Number of Data
/
Targets
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Citation
Author
Journal/Citation
Institution
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Special Data Sets
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PDB
85%
100%
Seq ID
UniProtKB/Swiss-Prot
UniProtKB/TrEMBL
PubMed
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All Compounds & Data
Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Targets Binding with 103 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
Abelson murine leukemia viral oncogene homolog 2
Ki:
2
IC50:
33
Kd:
145
20
11
2D
3D
TSV
Abelson-related gene protein
Ki:
2
IC50:
33
Kd:
145
20
11
2D
3D
TSV
ABL2
Ki:
2
IC50:
33
Kd:
145
20
11
2D
3D
TSV
EK4
IC50:
5
1
1
2D
3D
TSV
EPH-like kinase 4
IC50:
5
1
1
2D
3D
TSV
Epha3
IC50:
5
1
1
2D
3D
TSV
Etk1
IC50:
5
1
1
2D
3D
TSV
Leukocyte tyrosine kinase receptor
IC50:
22
Kd:
120
16
5
2D
3D
TSV
Mek4
IC50:
5
1
1
2D
3D
TSV
Mitogen-activated protein kinase kinase kinase 10
IC50:
22
Kd:
122
13
4
2D
3D
TSV
Mixed Lineage Kinase 2 (MLK2)
IC50:
22
Kd:
122
13
4
2D
3D
TSV
MLK2
IC50:
22
Kd:
122
13
4
2D
3D
TSV
Tyro4
IC50:
5
1
1
2D
3D
TSV
Tyrosine kinase ARG
Ki:
2
IC50:
33
Kd:
145
20
11
2D
3D
TSV
Tyrosine-protein kinase ABL2
Ki:
2
IC50:
33
Kd:
145
20
11
2D
3D
TSV
Tyrosine-protein kinase receptor ETK1
IC50:
5
Kd:
15
3
1
2D
3D
TSV
Tyrosine-protein kinase TYRO4
IC50:
5
Kd:
15
3
1
2D
3D
TSV