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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
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Het List in SDF
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Important Compounds
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Name
SMILES
Number of Data
/
Targets
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85%
100%
Seq ID
UniProtKB/Swiss-Prot
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Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Deposition
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Targets Binding with 226 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
2.7.12.2
Ki:
1
IC50:
233
4
7
2D
3D
TSV
Cancer/testis antigen 84
Ki:
1
IC50:
233
4
7
2D
3D
TSV
CT84
Ki:
1
IC50:
233
4
7
2D
3D
TSV
EcMetAP
IC50:
369
8
3
2D
3D
TSV
Lymphokine-activated killer T-cell-originated protein kinase
Ki:
1
IC50:
233
4
7
2D
3D
TSV
MAPKK-like protein kinase
Ki:
1
IC50:
233
4
7
2D
3D
TSV
Methionine aminopeptidase
IC50:
369
8
3
2D
3D
TSV
Nori-3
Ki:
1
IC50:
233
4
7
2D
3D
TSV
PBK
Ki:
1
IC50:
233
4
7
2D
3D
TSV
PDZ-binding kinase
Ki:
1
IC50:
233
4
7
2D
3D
TSV
Spermatogenesis-related protein kinase
Ki:
1
IC50:
233
4
7
2D
3D
TSV
SPK
Ki:
1
IC50:
233
4
7
2D
3D
TSV
T-LAK cell-originated protein kinase
Ki:
1
IC50:
233
4
7
2D
3D
TSV
TOPK
Ki:
1
IC50:
233
4
7
2D
3D
TSV