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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
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Important Compounds
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Name
SMILES
Number of Data
/
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85%
100%
Seq ID
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Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Targets Binding with 289 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
C-mpl
EC50:
327
10
3
2D
3D
TSV
CD_antigen=CD110
EC50:
327
10
3
2D
3D
TSV
Dual-specificity tyrosine-phosphorylation regulated kinase 2
IC50:
164
Kd:
81
23
4
2D
3D
TSV
Myeloproliferative leukemia protein
EC50:
327
10
3
2D
3D
TSV
P-selectin
IC50:
309
29
6
2D
3D
TSV
P-selectin/P-selectin glycoprotein ligand 1
IC50:
350
30
12
2D
3D
TSV
Prostaglandin E synthase 2
IC50:
296
6
6
2D
3D
TSV
Rac1 protein
Ki:
117
IC50:
18
EC50:
469
17
8
2D
3D
TSV
Ras-related C3 botulinum toxin substrate 1
Ki:
117
IC50:
18
EC50:
469
17
8
2D
3D
TSV
Ras-related C3 botulinum toxin substrate 1/T-lymphoma invasion and metastasis-inducing protein 1
Ki:
117
IC50:
18
EC50:
469
17
8
2D
3D
TSV
Thrombopoietin receptor
EC50:
327
10
3
2D
3D
TSV
TPO-R
EC50:
327
10
3
2D
3D
TSV