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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
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/
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Seq ID
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Ki
IC50
Kd
EC50
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ΔH°
-TΔS°
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Targets Binding with 47 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
Antigen p25
IC50:
47
Kd:
1
1
3
2D
3D
TSV
Arylamine N-acetyltransferase 1
IC50:
48
2
7
2D
3D
TSV
c-H-ras
IC50:
48
Kd:
2
5
7
2D
3D
TSV
Carbonic Anhydrase (hpCA)
Ki:
47
1
1
2D
3D
TSV
CBX5
IC50:
47
Kd:
1
1
3
2D
3D
TSV
CDY-like 2
IC50:
47
Kd:
1
1
3
2D
3D
TSV
CDYL2
IC50:
47
Kd:
1
1
3
2D
3D
TSV
Chromobox protein homolog 5
IC50:
47
Kd:
1
1
3
2D
3D
TSV
Chromodomain Y-like protein 2
IC50:
47
Kd:
1
1
3
2D
3D
TSV
G-protein coupled receptor 91
IC50:
53
1
5
2D
3D
TSV
GPR91
IC50:
47
1
4
2D
3D
TSV
GTPase HRas
IC50:
48
Kd:
2
5
7
2D
3D
TSV
GTPase HRas, N-terminally processed
IC50:
48
Kd:
2
5
7
2D
3D
TSV
H-Ras
IC50:
48
Kd:
2
5
7
2D
3D
TSV
H-Ras-1
IC50:
48
Kd:
2
5
7
2D
3D
TSV
Ha-Ras
IC50:
48
Kd:
2
5
7
2D
3D
TSV
Ha-Ras-CVLS
IC50:
48
Kd:
2
5
7
2D
3D
TSV
Heterochromatin protein 1 homolog alpha
IC50:
47
Kd:
1
1
3
2D
3D
TSV
His6-Ha-Ras-CVLS
IC50:
48
Kd:
2
5
7
2D
3D
TSV
HP1 alpha
IC50:
47
Kd:
1
1
3
2D
3D
TSV
HP1A
IC50:
47
Kd:
1
1
3
2D
3D
TSV
hpCA
Ki:
47
1
1
2D
3D
TSV
Human herpesvirus 1 protease
Ki:
9
IC50:
49
3
3
2D
3D
TSV
IKs producing slow voltage-gated potassium channel subunit alpha KvLQT1
IC50:
54
3
4
2D
3D
TSV
IRE1α
IC50:
79
1
0
2D
3D
TSV
KQT-like 1
IC50:
54
3
4
2D
3D
TSV
LPL
IC50:
71
4
6
2D
3D
TSV
NanoLuc luciferase (Nluc)
IC50:
47
1
1
2D
3D
TSV
P-selectin glycoprotein ligand 1
IC50:
47
3
9
2D
3D
TSV
p21ras
IC50:
48
Kd:
2
5
7
2D
3D
TSV
P2Y purinoceptor 1-like
IC50:
47
1
4
2D
3D
TSV
Potassium voltage-gated channel subfamily KQT member 1
IC50:
54
3
4
2D
3D
TSV
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4
IC50:
37
EC50:
9
4
3
2D
3D
TSV
Protein-tyrosine phosphatase 4A3
IC50:
54
9
5
2D
3D
TSV
Sialidase 4
Ki:
3
IC50:
61
7
5
2D
3D
TSV
Succinate receptor 1
IC50:
53
1
5
2D
3D
TSV
Sucnr1
IC50:
6
1
1
2D
3D
TSV
Tc14DM
Kd:
34
4
4
2D
3D
TSV
Transforming protein p21
IC50:
48
Kd:
2
5
7
2D
3D
TSV
Transforming protein p21/H-Ras-1
IC50:
48
Kd:
2
5
7
2D
3D
TSV
Wild-type Ha-Ras
IC50:
48
Kd:
2
5
7
2D
3D
TSV
Xaa-Pro dipeptidase
Ki:
5
IC50:
62
6
11
2D
3D
TSV