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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
26670264 73 Fragment-Based Discovery of 2-Aminoquinazolin-4(3H)-ones As Novel Class Nonpeptidomimetic Inhibitors of the Plasmepsins I, II, and IV.EBI Latvian Institute of Organic Synthesis
24900843 60 Plasmepsin inhibitory activity and structure-guided optimization of a potent hydroxyethylamine-based antimalarial hit.EBI Latvian Institute of Organic Synthesis
10669559 180 Protease inhibitors: current status and future prospects.EBI University of Queensland
19635672 35 alpha-Substituted norstatines as the transition-state mimic in inhibitors of multiple digestive vacuole malaria aspartic proteases.EBI Uppsala University
19328682 13 Expedient solid-phase synthesis of both symmetric and asymmetric diol libraries targeting aspartic proteases.EBI National University of Singapore
17149873 20 High antiplasmodial activity of novel plasmepsins I and II inhibitors.EBI University of Milan
16162010 78 Synthesis of malarial plasmepsin inhibitors and prediction of binding modes by molecular dynamics simulations.EBI Uppsala University
15974592 68 Design and synthesis of potent inhibitors of plasmepsin I and II: X-ray crystal structure of inhibitor in complex with plasmepsin II.EBI LinköPing University
31913032 86 Plasmepsin Inhibitors in Antimalarial Drug Discovery: Medicinal Chemistry and Target Validation (2000 to Present).EBI University of Zambia
30529637 76 Peptidomimetic plasmepsin inhibitors with potent anti-malarial activity and selectivity against cathepsin D.EBI Latvian Institute of Organic Synthesis
29636223 84 2-Aminoquinazolin-4(3H)-one based plasmepsin inhibitors with improved hydrophilicity and selectivity.EBI Latvian Institute of Organic Synthesis
15658851 42 Selective estrogen receptor modulators with conformationally restricted side chains. Synthesis and structure-activity relationship of ERalpha-selective tetrahydroisoquinoline ligands.BDB Novartis Pharmaceuticals
15689158 21 Novel transient receptor potential vanilloid 1 receptor antagonists for the treatment of pain: structure-activity relationships for ureas with quinoline, isoquinoline, quinazoline, phthalazine, quinoxaline, and cinnoline moieties.BDB Abbott Laboratories
18072720 30 Stereospecific high-affinity TRPV1 antagonists: chiral N-(2-Benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide analogues.BDB Seoul National University
12639546 30 Identification of a high-affinity phosphopeptide inhibitor of Stat3.BDB The University of Texas At Houston