The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
24359257 |
10 |
Optimization of furin inhibitors to protect against the activation of influenza hemagglutinin H5 and Shiga toxin.![EBI](/images/logo_chembl.png) |
Universit£ |
24350995 |
46 |
Design, synthesis, and structure-activity relationship studies of a potent PACE4 inhibitor.![EBI](/images/logo_chembl.png) |
Universit£ |
23126600 |
34 |
The Multi-Leu peptide inhibitor discriminates between PACE4 and furin and exhibits antiproliferative effects on prostate cancer cells.![EBI](/images/logo_chembl.png) |
Universit£ |
22682919 |
26 |
Furin inhibitors: importance of the positive formal charge and beyond.![EBI](/images/logo_chembl.png) |
Torrey Pines Institute For Molecular Studies |
21757345 |
34 |
New substrate analogue furin inhibitors derived from 4-amidinobenzylamide.![EBI](/images/logo_chembl.png) |
Philipps University Marburg |
21168329 |
47 |
New furin inhibitors based on weakly basic amidinohydrazones.![EBI](/images/logo_chembl.png) |
Philipps University Marburg |
20045647 |
35 |
Synthesis and optimization of thiadiazole derivatives as a novel class of substrate competitive c-Jun N-terminal kinase inhibitors.![EBI](/images/logo_chembl.png) |
Institute For Medical Research |
20038105 |
50 |
Potent inhibitors of furin and furin-like proprotein convertases containing decarboxylated P1 arginine mimetics.![EBI](/images/logo_chembl.png) |
Philipps University Marburg |
19282190 |
4 |
Discovery of 2-(5-nitrothiazol-2-ylthio)benzo[d]thiazoles as novel c-Jun N-terminal kinase inhibitors.![EBI](/images/logo_chembl.png) |
Institute For Medical Research |
18977558 |
18 |
Modeling the activity of furin inhibitors using artificial neural network.![EBI](/images/logo_chembl.png) |
Mahidol University |
17537721 |
289 |
Targeting host cell furin proprotein convertases as a therapeutic strategy against bacterial toxins and viral pathogens.![EBI](/images/logo_chembl.png) |
Institute For Medical Research |
27045975 |
34 |
Notch Antagonists: Potential Modulators of Cancer and Inflammatory Diseases.![EBI](/images/logo_chembl.png) |
Centre Hospitalier Universitaire Vaudois (Chuv) |
7562936 |
10 |
Synthesis of tight binding inhibitors and their action on the proprotein-processing enzyme furin.![EBI](/images/logo_chembl.png) |
Friedrich Miescher-Institut |
30501188 |
24 |
Improving the Selectivity of PACE4 Inhibitors through Modifications of the P1 Residue.![EBI](/images/logo_chembl.png) |
TBA |
30180568 |
54 |
Increasing C-Terminal Hydrophobicity Improves the Cell Permeability and Antiproliferative Activity of PACE4 Inhibitors against Prostate Cancer Cell Lines.![EBI](/images/logo_chembl.png) |
Universit£ |
28287731 |
150 |
Positional Scanning Identifies the Molecular Determinants of a High Affinity Multi-Leucine Inhibitor for Furin and PACE4.![EBI](/images/logo_chembl.png) |
University of Gdansk |
24612767 |
7 |
Discovery of novel secretory phospholipase A2 inhibitors using virtual screen.![BDB](/images/logo_bindingdb.png) |
Peking University |