The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
24411477 |
84 |
Carbamazepine derivatives with P2X4 receptor-blocking activity.![EBI](/images/logo_chembl.png) |
University of Bonn |
20045645 |
66 |
Discovery and optimization of RO-85, a novel drug-like, potent, and selective P2X3 receptor antagonist.![EBI](/images/logo_chembl.png) |
Roche Palo Alto |
23075067 |
98 |
N-substituted phenoxazine and acridone derivatives: structure-activity relationships of potent P2X4 receptor antagonists.![EBI](/images/logo_chembl.png) |
University of Bonn |
12213051 |
207 |
Purine and pyrimidine (P2) receptors as drug targets.![EBI](/images/logo_chembl.png) |
National Institute of Diabetes |
19231180 |
81 |
Identification and SAR of novel diaminopyrimidines. Part 1: The discovery of RO-4, a dual P2X(3)/P2X(2/3) antagonist for the treatment of pain.![EBI](/images/logo_chembl.png) |
Roche Palo Alto |
19231178 |
61 |
Identification and SAR of novel diaminopyrimidines. Part 2: The discovery of RO-51, a potent and selective, dual P2X(3)/P2X(2/3) antagonist for the treatment of pain.![EBI](/images/logo_chembl.png) |
Roche Palo Alto |
11462975 |
50 |
Structure-activity relationships of pyridoxal phosphate derivatives as potent and selective antagonists of P2X1 receptors.![EBI](/images/logo_chembl.png) |
National Institute of Diabetes and Digestive and Kidney Diseases |
32345019 |
134 |
Discovery and Structure Relationships of Salicylanilide Derivatives as Potent, Non-acidic P2X1 Receptor Antagonists.![EBI](/images/logo_chembl.png) |
University of Bonn |
27427902 |
93 |
Potent Suppressive Effects of 1-Piperidinylimidazole Based Novel P2X7 Receptor Antagonists on Cancer Cell Migration and Invasion.![EBI](/images/logo_chembl.png) |
Gwangju Institute of Science and Technology (Gist) |
30996785 |
44 |
Investigation on 2',3'-![EBI](/images/logo_chembl.png) |
University of Camerino |
31532206 |
26 |
Development of High-Throughput Fluorescent-Based Screens to Accelerate Discovery of P2X Inhibitors from Animal Venoms.![EBI](/images/logo_chembl.png) |
University of East Anglia |
31746599 |
78 |
Discovery and Characterization of the Potent and Selective P2X4 Inhibitor ![EBI](/images/logo_chembl.png) |
Bayer |
26460788 |
45 |
Novel Series of Dihydropyridinone P2X7 Receptor Antagonists.![EBI](/images/logo_chembl.png) |
Hoffmann-La Roche |
29649742 |
55 |
Synthesis and structure-activity relationships of quinolinone and quinoline-based P2X7 receptor antagonists and their anti-sphere formation activities in glioblastoma cells.![EBI](/images/logo_chembl.png) |
Gwangju Institute of Science and Technology (Gist) |
29805055 |
40 |
Pyrrolinone derivatives as a new class of P2X3 receptor antagonists. Part 1: Initial structure-activity relationship studies of a hit from a high throughput screening.![EBI](/images/logo_chembl.png) |
Shionogi |
8730754 |
7 |
Pharmacological profile of TP-680, a new cholecystokininA receptor antagonist.![BDB](/images/logo_bindingdb.png) |
University of Occupational and Environmental Health |