The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
28435528 |
24 |
Discovery of Highly Selective Inhibitors of the Immunoproteasome Low Molecular Mass Polypeptide 2 (LMP2) Subunit. |
Kezar Life Sciences |
25006746 |
85 |
Structure-based design of฿1i or฿5i specific inhibitors of human immunoproteasomes. |
Leiden Institute of Chemistry and Netherlands Proteomics Centre |
30380863 |
196 |
Required Immunoproteasome Subunit Inhibition Profile for Anti-Inflammatory Efficacy and Clinical Candidate KZR-616 ((2 S,3 R)- N-(( S)-3-(Cyclopent-1-en-1-yl)-1-(( R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-hydroxy-3-(4-methoxyphenyl)-2-(( S)-2-(2-morpholinoacetamido)propanamido)propenamide). |
Kezar Life Sciences |
31521028 |
67 |
Immunoproteasome-selective inhibitors: An overview of recent developments as potential drugs for hematologic malignancies and autoimmune diseases. |
Hangzhou Xixi Hospital |
30657666 |
263 |
Structure-Based Design of Inhibitors Selective for Human Proteasome ?2c or ?2i Subunits. |
Leiden Institute of Chemistry and Netherlands Proteomics Centre |
30455150 |
10 |
Tetradehydrohalicyclamine B, a new proteasome inhibitor from the marine sponge Acanthostrongylophora ingens. |
Kumamoto University |
29339252 |
124 |
Structure-based design of human immuno- and constitutive proteasomes inhibitors. |
Universit£ |
29782167 |
48 |
Potent and Highly Selective Inhibitors of the Proteasome Trypsin-like Site by Incorporation of Basic Side Chain Containing Amino Acid Derived Sulfonyl Fluorides. |
University of Glasgow |