The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 28131094 |
66 |
New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation. |
Universities of Lille |
| 26390077 |
42 |
Tactical Approaches to Interconverting GPCR Agonists and Antagonists. |
University of Minnesota |
| 26820449 |
84 |
Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives. |
Universit£ |
| 26785296 |
32 |
Synthesis of 2-arylfuro[3,2-b]pyridines: Effect of the C2-aryl group on melatoninergic activity. |
Universit£ |
| 26367450 |
4 |
New coumarin-based fluorescent melatonin ligands. Design, synthesis and pharmacological characterization. |
Iqm-Csic |
| 26023814 |
79 |
Novel N-Acetyl Bioisosteres of Melatonin: Melatonergic Receptor Pharmacology, Physicochemical Studies, and Phenotypic Assessment of Their Neurogenic Potential. |
Iqm-Csic |
| 25232966 |
52 |
Efficient synthesis of hexahydroindenopyridines and their potential as melatoninergic ligands. |
Universidad De Valencia |
| 24228714 |
64 |
MT1 and MT2 melatonin receptors: ligands, models, oligomers, and therapeutic potential. |
The German University In Cairo |
| 23228808 |
22 |
Development of substituted N-[3-(3-methoxylphenyl)propyl] amides as MT(2)-selective melatonin agonists: improving metabolic stability. |
Hong Kong University of Science and Technology |
| 23265885 |
30 |
Synthesis of new N-(arylcyclopropyl)acetamides and N-(arylvinyl)acetamides as conformationally-restricted ligands for melatonin receptors. |
Paris-Sud University |
| 21775151 |
22 |
Bivalent ligand approach on N-{2-[(3-methoxyphenyl)methylamino]ethyl}acetamide: synthesis, binding affinity and intrinsic activity for MT(1) and MT(2) melatonin receptors. |
Universit£ |
| 20674373 |
84 |
Design, synthesis, and pharmacological effects of structurally simple ligands for MT(1) and MT(2) melatonin receptors. |
Universit£ |
| 20444610 |
71 |
Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands. |
University of Lille |
| 10737738 |
78 |
Mapping the melatonin receptor. 6. Melatonin agonists and antagonists derived from 6H-isoindolo[2,1-a]indoles, 5,6-dihydroindolo[2,1-a]isoquinolines, and 6,7-dihydro-5H-benzo[c]azepino[2,1-a]indoles. |
King'S College London |
| 21764185 |
12 |
Design and synthesis of 2-phenylimidazo[1,2-a]pyridines as a novel class of melatonin receptor ligands. |
Universit£ |
| 21568291 |
30 |
Synthesis of a novel series of tricyclic dihydrofuran derivatives: discovery of 8,9-dihydrofuro[3,2-c]pyrazolo[1,5-a]pyridines as melatonin receptor (MT1/MT2) ligands. |
Takeda Pharmaceutical |
| 21392858 |
28 |
Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands. |
University of Lille |
| 21473625 |
42 |
1,6-Dihydro-2H-indeno[5,4-b]furan derivatives: design, synthesis, and pharmacological characterization of a novel class of highly potent MT2-selective agonists. |
Takeda Pharmaceutical |
| 21377769 |
30 |
Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3. |
University of Lille |
| 21420861 |
50 |
Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists. |
Universit£ |
| 20621473 |
56 |
Discovery of potent, selective, and orally bioavailable 3H-spiro[isobenzofuran-1,4'-piperidine] based melanocortin subtype-4 receptor agonists. |
Merck Research Laboratories |
| 20227878 |
40 |
Synthesis of substituted N-[3-(3-methoxyphenyl)propyl] amides as highly potent MT(2)-selective melatonin ligands. |
Hong Kong University of Science and Technology |
| 19473848 |
7 |
Synthesis and pharmacological evaluation of 1,2,3,4-tetrahydropyrazino[1,2-a]indole and 2-[(phenylmethylamino)methyl]-1H-indole analogues as novel melatoninergic ligands. |
University of W£Rzburg |
| | 26 |
The development of a charged melatonin receptor ligand |
TBA |
| | 12 |
Synthesis and receptor binding studies of quinolinic derivatives as melatonin receptor ligands |
TBA |
| 19193160 |
42 |
2-[(2,3-dihydro-1H-indol-1-yl)methyl]melatonin analogues: a novel class of MT2-selective melatonin receptor antagonists. |
University of WüRzburg |
| 18778943 |
53 |
Synthesis of 3-phenylnaphthalenic derivatives as new selective MT(2) melatoninergic ligands. |
University of Lille 2 |
| 18657980 |
14 |
Synthesis and pharmacological evaluation of pentacyclic 6a,7-dihydrodiindole and 2,3-dihydrodiindole derivatives as novel melatoninergic ligands. |
University of WüRzburg |
| 18372181 |
32 |
Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3. |
Université |
| 17481904 |
24 |
Synthesis and biological activity of new melatonin dimeric derivatives. |
Università |
| 16759094 |
70 |
Mapping the melatonin receptor. 7. Subtype selective ligands based on beta-substituted N-acyl-5-methoxytryptamines and beta-substituted N-acyl-5-methoxy-1-methyltryptamines. |
University of Athens |
| 15713384 |
28 |
(R)-2-(4-Phenylbutyl)dihydrobenzofuran derivatives as melatoninergic agents. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 15501061 |
51 |
Tetrahydroisoquinoline derivatives as melatonin MT2 receptor antagonists. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 15380218 |
40 |
N-[2-[2-(4-Phenylbutyl)benzofuran-4-yl]cyclopropylmethyl]acetamide: an orally bioavailable melatonin receptor agonist. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 15203165 |
80 |
Synthesis and structure-activity relationship of novel benzoxazole derivatives as melatonin receptor agonists. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 15013015 |
76 |
4-Substituted anilides as selective melatonin MT2 receptor agonists. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 14980664 |
48 |
Design and synthesis of benzoxazole derivatives as novel melatoninergic ligands. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 14643330 |
40 |
Heterocyclic aminopyrrolidine derivatives as melatoninergic agents. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 12646022 |
22 |
Design and synthesis of naphthalenic dimers as selective MT1 melatoninergic ligands. |
Université |
| 12643943 |
43 |
Indanyl piperazines as melatonergic MT2 selective agents. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 12213063 |
4 |
Synthesis of a novel series of tricyclic indan derivatives as melatonin receptor agonists. |
Takeda Chemical Industries |
| 12061881 |
94 |
Synthesis and structure-affinity-activity relationships of novel benzofuran derivatives as MT(2) melatonin receptor selective ligands. |
Institut De Chimie Pharmaceutique Albert Lespagnol |
| 11960497 |
36 |
Synthesis of nitroindole derivatives with high affinity and selectivity for melatoninergic binding sites MT(3). |
Institut De Chimie Pharmaceutique Albert Lespagnol |
| 11063602 |
84 |
Synthesis of phenalene and acenaphthene derivatives as new conformationally restricted ligands for melatonin receptors. |
Paris-Sud University |
| 31298539 |
18 |
Design, Synthesis, and Characterization of Ogerin-Based Positive Allosteric Modulators for G Protein-Coupled Receptor 68 (GPR68). |
Icahn School of Medicine At Mount Sinai |
| 31204226 |
4 |
Polybenzyls from Gastrodia elata, their agonistic effects on melatonin receptors and structure-activity relationships. |
Chinese Academy of Sciences |
| 9435890 |
7 |
Development of a high-affinity ligand that binds irreversibly to Mel1b melatonin receptors. |
Duquesne University |
| 31727472 |
30 |
Indole-based melatonin analogues: Synthetic approaches and biological activity. |
Nantong University |
| 24900790 |
8 |
Original Design of Fluorescent Ligands by Fusing BODIPY and Melatonin Neurohormone. |
Universit£ |
| 18052314 |
32 |
N-(substituted-anilinoethyl)amides: design, synthesis, and pharmacological characterization of a new class of melatonin receptor ligands. |
Universit£ |
| 17459711 |
55 |
7-Substituted-melatonin and 7-substituted-1-methylmelatonin analogues: effect of substituents on potency and binding affinity. |
University College London |
| 15943478 |
22 |
Analysis of structure-activity relationships for MT2 selective antagonists by melatonin MT1 and MT2 receptor models. |
Universit£ |
| 15293992 |
26 |
Tricyclic alkylamides as melatonin receptor ligands with antagonist or inverse agonist activity. |
Universit£ |
| 12672242 |
8 |
Three-dimensional quantitative structure-activity relationship studies on selected MT1 and MT2 melatonin receptor ligands: requirements for subtype selectivity and intrinsic activity modulation. |
Universit£ |
| 11520198 |
54 |
2-N-acylaminoalkylindoles: design and quantitative structure-activity relationship studies leading to MT2-selective melatonin antagonists. |
Universit£ |
| 30015074 |
2 |
Synthesis and biological evaluation of magnolol derivatives as melatonergic receptor agonists with potential use in depression. |
Chinese Academy of Sciences |
| 29102176 |
135 |
Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT |
Univ. Lille |
| 30126274 |
44 |
Identification of Bivalent Ligands with Melatonin Receptor Agonist and Fatty Acid Amide Hydrolase (FAAH) Inhibitory Activity That Exhibit Ocular Hypotensive Effect in the Rabbit. |
Universit£ |
| 29595267 |
39 |
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands. |
Universit£ |
| 27894776 |
26 |
Design, synthesis, cyclooxygenase inhibition and biological evaluation of new 1,3,5-triaryl-4,5-dihydro-1H-pyrazole derivatives possessing amino/methanesulfonyl pharmacophore. |
Beni-Suef University |
| 26398140 |
54 |
1-(4-Methane(amino)sulfonylphenyl)-3-(4-substituted-phenyl)-5-(4-trifluoromethylphenyl)-1H-2-pyrazolines/pyrazoles as potential anti-inflammatory agents. |
Beni-Suef University |
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