The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26101564 |
20 |
MLN8054 and Alisertib (MLN8237): Discovery of Selective Oral Aurora A Inhibitors. |
Takeda Pharmaceutical |
23121096 |
86 |
Ion channels as therapeutic targets: a drug discovery perspective. |
Pfizer |
22734650 |
6 |
Allyl m-trifluoromethyldiazirine mephobarbital: an unusually potent enantioselective and photoreactive barbiturate general anesthetic. |
Massachusetts General Hospital |
18537233 |
108 |
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit. |
Moltech |
21277199 |
29 |
Exploring subtype selectivity and metabolic stability of a novel series of ligands for the benzodiazepine binding site of the GABAA receptor. |
Novartis Institutes For Biomedical Research |
| 7 |
A conformational study of ligands for omega modulatory sites of GABAa receptors by NOESY NMR spectroscopy and distance geometry |
TBA |
17626010 |
4 |
Proximity-accelerated chemical coupling reaction in the benzodiazepine-binding site of gamma-aminobutyric acid type A receptors: superposition of different allosteric modulators. |
University of Bern |
17311911 |
2 |
Identification of anesthetic binding sites on human serum albumin using a novel etomidate photolabel. |
Imperial College |
12408715 |
97 |
Synthesis and biological evaluation of 7,8,9,10-tetrahydroimidazo[1,2-c]pyrido[3,4-e]pyrimdin-5(6H)-ones as functionally selective ligands of the benzodiazepine receptor site on the GABA(A) receptor. |
Neurogen |
31404862 |
138 |
Imidazopyridine-based selective and multifunctional ligands of biological targets associated with psychiatric and neurodegenerative diseases. |
Palack£ |
31738537 |
95 |
Subtype Selective ?-Aminobutyric Acid Type A Receptor (GABA |
University of Sussex |
28759875 |
30 |
An overview of benzo[b]thiophene-based medicinal chemistry. |
Jain University |
26833890 |
18 |
Synthesis, Biological Evaluation, and Molecular Docking of 8-imino-2-oxo-2H,8H-pyrano[2,3-f]chromene Analogs: New Dual AChE Inhibitors as Potential Drugs for the Treatment of Alzheimer's Disease. |
Yogi Vemana University |
26469307 |
7 |
Phosphorylation of Capsaicinoid Derivatives Provides Highly Potent and Selective Inhibitors of the Transcription Factor STAT5b. |
University of Leipzig |
26214255 |
11 |
The amylase inhibitor montbretin A reveals a new glycosidase inhibition motif. |
University of British Columbia |
25636004 |
12 |
Structure-guided design of a high affinity inhibitor to human CtBP. |
University of Massachusetts Medical School |