BindingDB logo
myBDB logout

17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
15013018 48 1,2-Benzothiazine 1,1-dioxide alpha-ketoamide analogues as potent calpain I inhibitors.EBI Cephalon
11055335 27 Highly potent and selective peptide-based inhibitors of the hepatitis C virus serine protease: towards smaller inhibitors.EBI Boehringer Ingelheim Pharmaceuticals
 24 Inhibition of human cytomegalovirus protease by benzoxazinones and evidence of antiviral activity in cell cultureEBI TBA
 1 Peptidyl epoxides as inhibitors of α-chymotrypsin: Remarkable change from irreversible to reversible competitive inhibitor as a consequence of the improvement of binding affinityEBI TBA
 4 Inactivation of serine protease, α-chymotrypsin by fluorinated phenylalanine analoguesEBI TBA
 6 N-(carbobenzyloxy)isatin: A slow binding α-keto lactam inhibitor of α-chymotrypsinEBI TBA
14741272 7 Inhibition of alpha-chymotrypsin with thiol-bearing substrate analogues in the presence of zinc ion.EBI Pohang University of Science and Technology
12668020 29 Oxyguanidines: application to non-peptidic phenyl-based thrombin inhibitors.EBI 3-Dimensional Pharmaceuticals
10328293 23 The discovery of orally available thrombin inhibitors: optimisation of the P1 pharmacophore.EBI Novartis Horsham Research Centre
10091694 90 Symmetrical anhydride-type serine protease inhibitors: structure-activity relationship studies of human chymase inhibitors.EBI Nippon Steel
9871780 85 Inhibition of human cytomegalovirus protease N(o) with monocyclic beta-lactams.EBI Boehringer Ingelheim (Canada)
9871680 5 Potent and selective inhibitors of the proteasome: dipeptidyl boronic acids.EBI Proscript
31413811 26 Iterative Optimization of the Cyclic Peptide SFTI-1 Yields Potent Inhibitors of Neutrophil Proteinase 3.EBI The University of Queensland
3851848 14 Acylamino boronic acids and difluoroborane analogues of amino acids: potent inhibitors of chymotrypsin and elastase.EBI TBA
3512826 3 Enol lactone inhibitors of serine proteases. The effect of regiochemistry on the inactivation behavior of phenyl-substituted (halomethylene)tetra- and -dihydrofuranones and (halomethylene)tetrahydropyranones toward alpha-chymotrypsin: stable acyl enzyme intermediate.EBI TBA
2296031 48 Synthesis of peptidyl fluoromethyl ketones and peptidyl alpha-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G.EBI Merrell Dow Research Institute