The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
15013018 |
48 |
1,2-Benzothiazine 1,1-dioxide alpha-ketoamide analogues as potent calpain I inhibitors. |
Cephalon |
11055335 |
27 |
Highly potent and selective peptide-based inhibitors of the hepatitis C virus serine protease: towards smaller inhibitors. |
Boehringer Ingelheim Pharmaceuticals |
| 24 |
Inhibition of human cytomegalovirus protease by benzoxazinones and evidence of antiviral activity in cell culture |
TBA |
| 1 |
Peptidyl epoxides as inhibitors of α-chymotrypsin: Remarkable change from irreversible to reversible competitive inhibitor as a consequence of the improvement of binding affinity |
TBA |
| 4 |
Inactivation of serine protease, α-chymotrypsin by fluorinated phenylalanine analogues |
TBA |
| 6 |
N-(carbobenzyloxy)isatin: A slow binding α-keto lactam inhibitor of α-chymotrypsin |
TBA |
14741272 |
7 |
Inhibition of alpha-chymotrypsin with thiol-bearing substrate analogues in the presence of zinc ion. |
Pohang University of Science and Technology |
12668020 |
29 |
Oxyguanidines: application to non-peptidic phenyl-based thrombin inhibitors. |
3-Dimensional Pharmaceuticals |
10328293 |
23 |
The discovery of orally available thrombin inhibitors: optimisation of the P1 pharmacophore. |
Novartis Horsham Research Centre |
10091694 |
90 |
Symmetrical anhydride-type serine protease inhibitors: structure-activity relationship studies of human chymase inhibitors. |
Nippon Steel |
9871780 |
85 |
Inhibition of human cytomegalovirus protease N(o) with monocyclic beta-lactams. |
Boehringer Ingelheim (Canada) |
9871680 |
5 |
Potent and selective inhibitors of the proteasome: dipeptidyl boronic acids. |
Proscript |
3851848 |
14 |
Acylamino boronic acids and difluoroborane analogues of amino acids: potent inhibitors of chymotrypsin and elastase. |
TBA |
3512826 |
3 |
Enol lactone inhibitors of serine proteases. The effect of regiochemistry on the inactivation behavior of phenyl-substituted (halomethylene)tetra- and -dihydrofuranones and (halomethylene)tetrahydropyranones toward alpha-chymotrypsin: stable acyl enzyme intermediate. |
TBA |
2296031 |
48 |
Synthesis of peptidyl fluoromethyl ketones and peptidyl alpha-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G. |
Merrell Dow Research Institute |