The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27128184 |
13 |
Design, synthesis and biological evaluation of PSMA/hepsin-targeted heterobivalent ligands. |
Korea University |
26985294 |
114 |
Design and Synthesis of Nonpeptide Inhibitors of Hepatocyte Growth Factor Activation. |
Southern Research |
26711145 |
24 |
Structure-based design, synthesis, and biological evaluation of Leu-Arg dipeptide analogs as novel hepsin inhibitors. |
Korea University |
26421993 |
44 |
Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors. |
Aurigene Discovery Technologies |
25882520 |
64 |
Structure-based discovery of small molecule hepsin and HGFA protease inhibitors: Evaluation of potency and selectivity derived from distinct binding pockets. |
Washington University |
25408834 |
63 |
Inhibitors of HGFA, Matriptase, and Hepsin Serine Proteases: A Nonkinase Strategy to Block Cell Signaling in Cancer. |
Washington University |
24900505 |
11 |
Design and synthesis of potent, selective inhibitors of matriptase. |
TBA |
30571119 |
67 |
Discovery of Selective Matriptase and Hepsin Serine Protease Inhibitors: Useful Chemical Tools for Cancer Cell Biology. |
Washington University School of Medicine |
30904782 |
12 |
Multi-target compounds acting in cancer progression: Focus on thiosemicarbazone, thiazole and thiazolidinone analogues. |
Universidade Federal De Pernambuco |
29701962 |
83 |
Design, Synthesis, and Testing of Potent, Selective Hepsin Inhibitors via Application of an Automated Closed-Loop Optimization Platform. |
University of Helsinki |