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25 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
24654918 19 Pharmacophoric modifications lead to superpotentavß3 integrin ligands with suppresseda5ß1 activity.EBI Technische Universit£T M£Nchen
23362923 59 Biselectivity of isoDGR peptides for fibronectin binding integrin subtypesa5ß1 andavß6: conformational control through flanking amino acids.EBI Technische Universit£T M£Nchen
17399986 114 R-isomers of Arg-Gly-Asp (RGD) mimics as potent alphavbeta3 inhibitors.EBI Pfizer
17387018 74 Discovery of +(2-{4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]phenyl}-cyclopropyl)acetic acid as potent and selective alphavbeta3 inhibitor: design, synthesis, and optimization.EBI Pfizer
16621534 87 Synthesis of pyrazoles and isoxazoles as potent alpha(v)beta3 receptor antagonists.EBI Pfizer
16303301 44 Synthesis of 2,5-thiazole butanoic acids as potent and selective alpha(v)beta3 integrin receptor antagonists with improved oral pharmacokinetic properties.EBI Pfizer
16298127 80 Convergent, parallel synthesis of a series of beta-substituted 1,2,4-oxadiazole butanoic acids as potent and selective alpha(v)beta3 receptor antagonists.EBI Pfizer
11855984 102 Nanomolar small molecule inhibitors for alphav(beta)6, alphav(beta)5, and alphav(beta)3 integrins.EBI Merck
32094009 36 Novel cilengitide-based cyclic RGD peptides as ?v?EBI Division of Organic Chemistry Csir-National Chemical Laboratory (Ncl)
30657681 262 Selective Targeting of Integrin ?v?8 by a Highly Active Cyclic Peptide.EBI Technische Universit£T M£Nchen
31381331 70 Profile of a Highly Selective Quaternized Pyrrolidine Betaine ?EBI Glaxosmithkline Medicines Research Centre
31497959 48 Discovery of an Orally Bioavailable Pan ?v Integrin Inhibitor for Idiopathic Pulmonary Fibrosis.EBI Glaxosmithkline Medicines Research Centre
24568695 76 Strategies to inhibit tumor associated integrin receptors: rationale for dual and multi-antagonists.EBI University of Bradford
25408832 152 Structure Activity Relationships of ?v Integrin Antagonists for Pulmonary Fibrosis by Variation in Aryl Substituents.EBI University of Nottingham
30215258 228 Discovery of ( S)-3-(3-(3,5-Dimethyl-1 H-pyrazol-1-yl)phenyl)-4-(( R)-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-yl)butanoic Acid, a Nonpeptidic ?EBI University of Strathclyde