The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
32143887 |
58 |
Design and synthesis of novel 2-arylbenzimidazoles as selective mutant isocitrate dehydrogenase 2 R140Q inhibitors. |
Shandong Provincial Hospital Affiliated To Shandong University |
31199148 |
148 |
Discovery and Optimization of Quinolinone Derivatives as Potent, Selective, and Orally Bioavailable Mutant Isocitrate Dehydrogenase 1 (mIDH1) Inhibitors. |
Forma Therapeutics |
32071674 |
30 |
Vorasidenib (AG-881): A First-in-Class, Brain-Penetrant Dual Inhibitor of Mutant IDH1 and 2 for Treatment of Glioma. |
Agios Pharmaceuticals |
30600148 |
65 |
Synthesis and biological evaluation of 3-aryl-4-indolyl-maleimides as potent mutant isocitrate dehydrogenase-1 inhibitors. |
Zhejiang University |
31971798 |
40 |
Structure-Based Design and Identification of FT-2102 (Olutasidenib), a Potent Mutant-Selective IDH1 Inhibitor. |
Forma Therapeutics |
29847930 |
142 |
Inhibitors of Mutant Isocitrate Dehydrogenases 1 and 2 (mIDH1/2): An Update and Perspective. |
China Pharmaceutical University |
29079473 |
62 |
Discovery and structure-activity-relationship study of novel conformationally restricted indane analogues for mutant isocitric dehydrogenase 1 (IDH1) inhibitors. |
Shanghai Haihe |
29057059 |
82 |
Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII. |
Saint Petersburg State University |
17293454 |
7 |
An in vitro and in vivo disconnect uncovered through high-throughput identification of botulinum neurotoxin A antagonists. |
The Scripps Research Institute |