The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27658368 |
54 |
Design and synthesis of selective, dual fatty acid binding protein 4 and 5 inhibitors. |
F. Hoffmann-La Roche |
27460668 |
18 |
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation. |
Chinese Academy of Sciences |
27096055 |
5 |
Interaction Analysis of FABP4 Inhibitors by X-ray Crystallography and Fragment Molecular Orbital Analysis. |
Ajinomoto |
25461324 |
18 |
Novel fatty acid binding protein 4 (FABP4) inhibitors: virtual screening, synthesis and crystal structure determination. |
Chinese Academy of Sciences |
23395658 |
49 |
Structure-guided design, synthesis and in vitro evaluation of a series of pyrazole-based fatty acid binding protein (FABP) 3 ligands. |
Okayama University 1-1-1 |
12036355 |
36 |
Simple, intuitive calculations of free energy of binding for protein-ligand complexes. 1. Models without explicit constrained water. |
University of Parma |
21481589 |
14 |
New aromatic substituted pyrazoles as selective inhibitors of human adipocyte fatty acid-binding protein. |
Chinese Academy of Sciences |
20471252 |
22 |
Discovery of highly selective inhibitors of human fatty acid binding protein 4 (FABP4) by virtual screening. |
Chinese Academy of Sciences |
19754198 |
5 |
Identification and characterization of a small molecule inhibitor of Fatty Acid binding proteins. |
University of Minnesota |
19217286 |
45 |
N-Benzyl-indolo carboxylic acids: Design and synthesis of potent and selective adipocyte fatty-acid binding protein (A-FABP) inhibitors. |
Biovitrum |
17502136 |
66 |
Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP). |
Bristol-Myers Squibb Pharmaceutical Research Institute |
16884313 |
9 |
NMR structure of a potent small molecule inhibitor bound to human keratinocyte fatty acid-binding protein. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
15357970 |
26 |
Substituted benzylamino-6-(trifluoromethyl)pyrimidin-4(1H)-ones: a novel class of selective human A-FABP inhibitors. |
Biovitrum |
15357969 |
45 |
Discovery of inhibitors of human adipocyte fatty acid-binding protein, a potential type 2 diabetes target. |
Biovitrum |
32202425 |
47 |
Exploration of Fragment Binding Poses Leading to Efficient Discovery of Highly Potent and Orally Effective Inhibitors of FABP4 for Anti-inflammation. |
Chinese Academy of Sciences |
30703745 |
8 |
1,2,4-Triazolo[1,5-a]pyrimidines in drug design. |
University of California |
31420256 |
52 |
Identification of new dual FABP4/5 inhibitors based on a naphthalene-1-sulfonamide FABP4 inhibitor. |
Fudan University |
29775936 |
51 |
From hit to lead: Structure-based discovery of naphthalene-1-sulfonamide derivatives as potent and selective inhibitors of fatty acid binding protein 4. |
Fudan University |
18456494 |
19 |
Synthesis and structure based optimization of novel Akt inhibitors. |
Pfizer |
12113830 |
13 |
Inhibition of Src kinase activity by 4-anilino-7-thienyl-3-quinolinecarbonitriles. |
Wyeth Research |