The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
24900651 |
50 |
Irreversible inhibitors of cysteine proteases. |
Dart Neuroscience |
19715320 |
87 |
Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
University of Florida |
18366176 |
7 |
Identification of promiscuous small molecule activators in high-throughput enzyme activation screens. |
University of Illinois |
21903398 |
88 |
Exploiting differences in caspase-2 and -3 S2 subsites for selectivity: structure-based design, solid-phase synthesis and in vitro activity of novel substrate-based caspase-2 inhibitors. |
Chdi Management |
17181147 |
10 |
Synthesis of novel caspase inhibitors for characterization of the active caspase proteome in vitro and in vivo. |
University of Edinburgh |
15686936 |
210 |
Novel pyrazinone mono-amides as potent and reversible caspase-3 inhibitors. |
Merck Frosst Centre For Therapeutic Research |
27563406 |
128 |
Discovery of Fluoromethylketone-Based Peptidomimetics as Covalent ATG4B (Autophagin-1) Inhibitors. |
Roche Pharma Research and Early Development |
28615111 |
24 |
Synthesis and antitumor activities of 1,2,3-triazines and their benzo- and heterofused derivatives. |
Universit£ |
18308563 |
39 |
Probing the elusive catalytic activity of vertebrate class IIa histone deacetylases. |
Irbm/Merck Research Laboratories |
17685602 |
33 |
Discovery of 3,3'-(2,4-diaminopteridine-6,7-diyl)diphenol as an isozyme-selective inhibitor of PI3K for the treatment of ischemia reperfusion injury associated with myocardial infarction. |
Targegen |
14698155 |
68 |
Synthesis and evaluation of indenopyrazoles as cyclin-dependent kinase inhibitors. Part 4: Heterocycles at C3. |
Bristol-Myers Squibb |