The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
8809160 |
132 |
Design, synthesis, and evaluation of 2 beta-alkenyl penam sulfone acids as inhibitors of beta-lactamases. |
F. Hoffmann-La Roche |
21676616 |
15 |
Side chain SAR of bicyclicß-lactamase inhibitors (BLIs). 2. N-Alkylated and open chain analogs of MK-8712. |
Merck Research Labs |
21664132 |
47 |
Thiophenyl oxime-derived phosphonates as nano-molar class C beta-lactamase inhibitors reducing MIC of imipenem against Pseudomonas aeruginosa and Acinetobacter baumannii. |
Merck |
20921316 |
10 |
Mechanistic studies of the inactivation of TEM-1 and P99 by NXL104, a novel non-beta-lactam beta-lactamase inhibitor. |
Novexel |
20299220 |
4 |
4,7-Dichloro benzothien-2-yl sulfonylaminomethyl boronic acid: first boronic acid-derived beta-lactamase inhibitor with class A, C, and D activity. |
Merck |
20044254 |
14 |
Side chain SAR of bicyclic beta-lactamase inhibitors (BLIs). 1. Discovery of a class C BLI for combination with imipinem. |
Merck Research Labs |
9767633 |
76 |
Structure-based design of beta-lactamase inhibitors. 1. Synthesis and evaluation of bridged monobactams. |
F. Hoffmann-La Roche |
8064298 |
9 |
SB-202742, a novel beta-lactamase inhibitor isolated from Spondias mombin. |
Smithkline Beecham Pharmaceuticals |
8421286 |
44 |
Inhibitors of protein kinase C. 3. Potent and highly selective bisindolylmaleimides by conformational restriction. |
Roche Products |