The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27214509 |
1 |
Synthesis, characterization and antitubercular activities of novel pyrrolyl hydrazones and their Cu-complexes. |
S.E.T'S College of Pharmacy |
25461892 |
25 |
Piperazine derivatives: synthesis, inhibition of the Mycobacterium tuberculosis enoyl-acyl carrier protein reductase and SAR studies. |
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul |
25282650 |
8 |
Development of benzo[d]oxazol-2(3H)-ones derivatives as novel inhibitors of Mycobacterium tuberculosis InhA. |
Birla Institute of Technology |
24967731 |
2 |
Diarylthiazole: an antimycobacterial scaffold potentially targeting PrrB-PrrA two-component system. |
Astrazeneca |
25221657 |
3 |
2-Phenylindole and Arylsulphonamide: Novel Scaffolds Bactericidal against Mycobacterium tuberculosis. |
Astrazeneca |
25218910 |
16 |
Development of 2-(4-oxoquinazolin-3(4H)-yl)acetamide derivatives as novel enoyl-acyl carrier protein reductase (InhA) inhibitors for the treatment of tuberculosis. |
Birla Institute of Technology |
24450589 |
64 |
Encoded library technology as a source of hits for the discovery and lead optimization of a potent and selective class of bactericidal direct inhibitors of Mycobacterium tuberculosis InhA. |
Glaxosmithkline |
24107081 |
17 |
Methyl-thiazoles: a novel mode of inhibition with the potential to develop novel inhibitors targeting InhA in Mycobacterium tuberculosis. |
Astrazeneca India |
23314046 |
3 |
Identification of novel antimycobacterial chemical agents through the in silico multi-conformational structure-based drug screening of a large-scale chemical library. |
Kyushu Institute of Technology |
22483635 |
1 |
Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents. |
Cnrs |
18457948 |
27 |
Synthesis and in vitro antimycobacterial activity of B-ring modified diaryl ether InhA inhibitors. |
Stony Brook University |
20855214 |
6 |
2-Hexadecynoic acid inhibits plasmodial FAS-II enzymes and arrests erythrocytic and liver stage Plasmodium infections. |
University of London |
19428156 |
30 |
Discovery of potential new InhA direct inhibitors based on pharmacophore and 3D-QSAR analysis followed by in silico screening. |
China Pharmaceutical University |
18393405 |
1 |
Natural products, small molecules, and genetics in tuberculosis drug development. |
National Institute of Diabetes and Digestive and Kidney Diseases |
12141869 |
2 |
Agonodepsides a and B: two new depsides from a filamentous fungus F7524. |
Institute of Molecular and Cell Biology |
17560106 |
1 |
Synthesis of 4-phenoxybenzamide adenine dinucleotide as NAD analogue with inhibitory activity against enoyl-ACP reductase (InhA) of Mycobacterium tuberculosis. |
University of Minnesota |
30846404 |
34 |
Discovery and development of novel rhodanine derivatives targeting enoyl-acyl carrier protein reductase. |
Nanjing University |
32240584 |
7 |
Fragment-Based Design of |
University of Cambridge |
31227345 |
1 |
Discovery of novel N-methyl carbazole tethered rhodanine derivatives as direct inhibitors of Mycobacterium tuberculosis InhA. |
University of Kwazulu-Natal (Ukzn) |
31904960 |
8 |
Synthesis and Structure-Activity Relationship Studies of C2-Modified Analogs of the Antimycobacterial Natural Product Pyridomycin. |
Eth Zurich |
24900646 |
2 |
Synthesis and antimycobacterial activity of 2,1'-dihydropyridomycins. |
Swiss Federal Institute of Technology (Eth) Zurich |
29407960 |
67 |
An overview on crystal structures of InhA protein: Apo-form, in complex with its natural ligands and inhibitors. |
Cnrs |
28818767 |
2 |
Recent advances of pyrazole-containing derivatives as anti-tubercular agents. |
Wuhan University of Science and Technology |
29748048 |
3 |
Discovery of novel anti-tuberculosis agents with pyrrolo[1,2-a]quinoxaline-based scaffold. |
West China Hospital |
2188581 |
23 |
Muscarinic receptor subtypes. |
National Institute For Medical Research |