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27 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
26850376 36 Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors.EBI Kyoto University
26762835 342 Discovery of 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one (7ao) as a potent selective inhibitor of Polo like kinase 2 (PLK2).EBI Icahn School of Medicine At Mount Sinai
24359159 60 Discovery of 1-methyl-1H-imidazole derivatives as potent Jak2 inhibitors.EBI Astrazeneca
22339433 48 Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds.EBI Kyoto University
22726925 216 Discovery of 5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-(tert-butyl)pyridine-3-sulfonamide (CZC24758), as a potent, orally bioavailable and selective inhibitor of PI3K for the treatment of inflammatory disease.EBI Cellzome
18183025 12060 A quantitative analysis of kinase inhibitor selectivity.EBI Ambit Biosciences
8824261 8 Crystal structures of catalytic subunit of cAMP-dependent protein kinase in complex with isoquinolinesulfonyl protein kinase inhibitors H7, H8, and H89. Structural implications for selectivity.EBI Institute For Biochemistry
22115617 64 CK2a and CK2a' subunits differ in their sensitivity to 4,5,6,7-tetrabromo- and 4,5,6,7-tetraiodo-1H-benzimidazole derivatives.EBI The John Paul Ii Catholic University of Lublin
22037378 31824 Comprehensive analysis of kinase inhibitor selectivity.EBI Ambit Biosciences
19654408 2521 AC220 is a uniquely potent and selective inhibitor of FLT3 for the treatment of acute myeloid leukemia (AML).EBI Ambit Biosciences
32589844 3 Structural and Mechanistic Basis of the Inhibitory Potency of Selected 2-Aminothiazole Compounds on Protein Kinase CK2.EBI Universit£T Zu K£Ln
31757666 314 Discovery and optimization of heteroaryl piperazines as potent and selective PI3K? inhibitors.EBI Merck
30763817 39 Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach.EBI University of Naples Federico Ii
30384048 365 ASR352, A potent anticancer agent: Synthesis, preliminary SAR, and biological activities against colorectal cancer bulk, 5-fluorouracil/oxaliplatin resistant and stem cells.EBI University of Florida
24900617 2 Inhibition of CK2: An Attractive Therapeutic Target for Cancer Treatment.EBI Therachem Research Medilab (India)
22169261 38 Synthesis and SAR of inhibitors of protein kinase CK2: novel tricyclic quinoline analogs.EBI Cylene Pharmaceuticals
29945794 193 ROCK inhibitors 2. Improving potency, selectivity and solubility through the application of rationally designed solubilizing groups.EBI Vertex Pharmaceuticals
22299586 14 Inhibitory effect of novel pyrazole carboxamide derivatives on human carbonic anhydrase enzyme.BDB Dumlupinar University
21381887 3 Synthesis and biological evaluation of fused oxepinocoumarins as free radicals scavengers.BDB Aristotle University of Thessaloniki
 46 UROKINASE in CSAR_FULL_RELEASE_3JULY2012BDB Csar