The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
10753476 |
84 |
Phosphinic derivatives as new dual enkephalin-degrading enzyme inhibitors: synthesis, biological properties, and antinociceptive activities. |
University of Paris |
10602705 |
82 |
Investigation of subsite preferences in aminopeptidase A (EC 3.4.11.7) led to the design of the first highly potent and selective inhibitors of this enzyme. |
University of Paris |
8632427 |
80 |
Optimal recognition of neutral endopeptidase and angiotensin-converting enzyme active sites by mercaptoacyldipeptides as a means to design potent dual inhibitors. |
University of Paris |
8691458 |
60 |
Design of orally active dual inhibitors of neutral endopeptidase and angiotensin-converting enzyme with long duration of action. |
University of Paris |
7783143 |
66 |
Hydroxamic acids as potent inhibitors of endothelin-converting enzyme from human bronchiolar smooth muscle. |
Berlex Laboratories |
8021926 |
41 |
New thiol inhibitors of neutral endopeptidase EC 3.4.24.11: synthesis and enzyme active-site recognition. |
University of Paris |
2585440 |
34 |
Enkephalinase inhibitors. 1. 2,4-Dibenzylglutaric acid derivatives. |
Ciba-Geigy |
2900898 |
14 |
Retro-inverso concept applied to the complete inhibitors of enkephalin-degrading enzymes. |
Ua 498 Cnrs |
| 38 |
Kelatorphan and related analogs: potent and selective inhibitors of leukotriene A4 hydrolase |
TBA |
17070062 |
16 |
Novel selective inhibitors of neutral endopeptidase for the treatment of female sexual arousal disorder. |
Pfizer |
16821800 |
96 |
Novel selective inhibitors of neutral endopeptidase for the treatment of female sexual arousal disorder. Synthesis and activity of functionalized glutaramides. |
Pfizer |
12113828 |
63 |
N-[2-(Indan-1-yl)-3-mercapto-propionyl] amino acids as highly potent inhibitors of the three vasopeptidases (NEP, ACE, ECE): In vitro and In vivo activities. |
University of Paris |
8421293 |
32 |
Exploration of neutral endopeptidase active site by a series of new thiol-containing inhibitors. |
University of Paris |
8057292 |
83 |
Mercaptoacyl amino acid inhibitors of atriopeptidase. 1. Structure-activity relationship studies of methionine and S-alkylcysteine derivatives. |
Schering-Plough Research Institute |
2738884 |
30 |
New kelatorphan-related inhibitors of enkephalin metabolism: improved antinociceptive properties. |
University of Paris |
2522989 |
14 |
Carboxyalkyl dipeptides with atrial natriuretic factor potentiating and antihypertensive activity. |
Schering-Plough Research Institute |