BindingDB logo
myBDB logout

43 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
12639555 10 Synthesis and anti-influenza evaluation of orally active bicyclic ether derivatives related to zanamivir.EBI Sankyo
12113810 20 Synthesis and anti-influenza virus activity of 7-O-alkylated derivatives related to zanamivir.EBI Sankyo
12113809 12 Synthesis and anti-influenza virus activity of 4-guanidino-7-substituted Neu5Ac2en derivatives.EBI Sankyo
22677529 3 Pyrrolidinobenzoic acid inhibitors of influenza virus neuraminidase: the hydrophobic side chain influences type A subtype selectivity.EBI University of Alabama At Birmingham
18694948 17 Limited inhibitory effects of oseltamivir and zanamivir on human sialidases.EBI Miyagi Cancer Center Research Institute
15214773 76 Fragment-based drug discovery.EBI Sunesis Pharmaceuticals
11000002 10 BCX-1812 (RWJ-270201): discovery of a novel, highly potent, orally active, and selective influenza neuraminidase inhibitor through structure-based drug design.EBI Biocryst Pharmaceuticals
10602699 15 Binding constants of neuraminidase inhibitors: An investigation of the linear interaction energy method.EBI University of Southampton
9526556 18 Dihydropyrancarboxamides related to zanamivir: a new series of inhibitors of influenza virus sialidases. 2. Crystallographic and molecular modeling study of complexes of 4-amino-4H-pyran-6-carboxamides and sialidase from influenza virus types A and B.EBI Glaxo Wellcome Research and Development
8126701 3 Molecular modeling studies on ligand binding to sialidase from influenza virus and the mechanism of catalysis.EBI Monash University
11266166 36 Sialidase inhibitors related to zanamivir. Further SAR studies of 4-amino-4H-pyran-2-carboxylic acid-6-propylamides.EBI Glaxowellcome Medicines Research Centre
 22 Novel inhibitors of influenza sialidases related to zanamivir. Heterocyclic replacements of the glycerol sidechainEBI TBA
 51 Novel inhibitors of influenza sialidases related to GG167 structure-activity, crystallographic and Molecular dynamics studies with 4H-pyran-2-carboxylic acid 6-carboxamidesEBI TBA
 16 Novel inhibitors of influenza sialidase related to GG167 Synthesis of 4-amino and guanidino-4H-pyran-2-carboxylic acid-6-propylamides; selective inhibitors of influenza a virus sialidaseEBI TBA
22100261 12 Synthesis and biological evaluation of sialic acid derivatives containing a long hydrophobic chain at the anomeric position and their C-5 linked polymers as potent influenza virus inhibitors.EBI Saitama University
21843936 35 3D QSAR and docking study of flavone derivatives as potent inhibitors of influenza H1N1 virus neuraminidase.EBI Chinese Academy of Medical Sciences
20014777 6 Antiviral potential and molecular insight into neuraminidase inhibiting diarylheptanoids from Alpinia katsumadai.EBI University of Innsbruck
15828835 6 Dimeric zanamivir conjugates with various linking groups are potent, long-lasting inhibitors of influenza neuraminidase including H5N1 avian influenza.EBI Glaxosmithkline
15582424 6 Design, synthesis, and structural analysis of inhibitors of influenza neuraminidase containing a 2,3-disubstituted tetrahydrofuran-5-carboxylic acid core.EBI Abbott Laboratories
11312919 22 Design, synthesis, and structural analysis of influenza neuraminidase inhibitors containing pyrrolidine cores.EBI Abbott Laboratories
31744778 11 Design, synthesis and biological evaluation of substituted flavones and aurones as potential anti-influenza agents.EBI Prin. K.M. Kundnani College of Pharmacy
30576902 36 Boronate, trifluoroborate, sulfone, sulfinate and sulfonate congeners of oseltamivir carboxylic acid: Synthesis and anti-influenza activity.EBI National Taiwan University
31835169 68 Discovery of novel 1,2,3-triazole oseltamivir derivatives as potent influenza neuraminidase inhibitors targeting the 430-cavity.EBI Shandong University
10395473 19 Potent inhibition of influenza sialidase by a benzoic acid containing a 2-pyrrolidinone substituent.EBI University of Alabama At Birmingham
31324565 12 Total synthesis of dryocrassin ABBA and its analogues with potential inhibitory activity against drug-resistant neuraminidases.EBI Chinese Academy of Sciences
31176096 44 Design, synthesis and biological evaluation of "Multi-Site"-binding influenza virus neuraminidase inhibitors.EBI Shandong University
31128993 22 Investigation of flexibility of neuraminidase 150-loop using tamiflu derivatives in influenza A viruses H1N1 and H5N1.EBI Charles University
31857844 1 Discovery of Novel Neuraminidase Inhibitors by Structure-Based Virtual Screening, Structural Optimization, and Bioassay.EBI Shanghai Institute of Technology
31708183 3 Design, synthesis and biological evaluation of oseltamivir derivatives containing pyridyl group as potent inhibitors of neuraminidase for influenza A.EBI Wuyi University
23411074 2 Aspulvinones from a mangrove rhizosphere soil-derived fungus Aspergillus terreus Gwq-48 with anti-influenza A viral (H1N1) activity.EBI Ocean University of China
20116898 52 QSAR study of flavonoids and biflavonoids as influenza H1N1 virus neuraminidase inhibitors.EBI Universidad De Buenos Aires
29107426 16 Synthesis and biological evaluation of NHEBI Shenyang Pharmaceutical University
29198893 3 Synthesis and anti-influenza virus evaluation of triterpene-sialic acid conjugates.EBI Meiji Pharmaceutical University
28958846 24 Discovery of berberine based derivatives as anti-influenza agent through blocking of neuraminidase.EBI Konkuk University
29965752 158 Optimization of N-Substituted Oseltamivir Derivatives as Potent Inhibitors of Group-1 and -2 Influenza A Neuraminidases, Including a Drug-Resistant Variant.EBI Shandong University
28984452 6 C-Methylated Flavonoid Glycosides from Pentarhizidium orientale Rhizomes and Their Inhibitory Effects on the H1N1 Influenza Virus.EBI Seoul National University
16621549 40 Novel 5-azaindole factor VIIa inhibitors.BDB Celera
14561087 27 Structure-activity relationships of the p38alpha MAP kinase inhibitor 1-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)naph- thalen-1-yl]urea (BIRB 796).BDB Boehringer Ingelheim Pharmaceuticals
11896401 3 Inhibition of p38 MAP kinase by utilizing a novel allosteric binding site.BDB Boehringer Ingelheim Pharmaceuticals
15857116 5 1-(5-Chloro-2-alkoxyphenyl)-3-(5-cyanopyrazin-2-yl)ureas [correction of cyanopyrazi] as potent and selective inhibitors of Chk1 kinase: synthesis, preliminary SAR, and biological activities.BDB Abbott Laboratories
16303309 31 Bicyclic and tricyclic thiophenes as protein tyrosine phosphatase 1B inhibitors.BDB Wyeth Research
10694412 15 Thermodynamics of substrate binding to the chaperone SecB.BDB Indian Institute of Science