The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
12639555 |
10 |
Synthesis and anti-influenza evaluation of orally active bicyclic ether derivatives related to zanamivir. |
Sankyo |
12113810 |
20 |
Synthesis and anti-influenza virus activity of 7-O-alkylated derivatives related to zanamivir. |
Sankyo |
12113809 |
12 |
Synthesis and anti-influenza virus activity of 4-guanidino-7-substituted Neu5Ac2en derivatives. |
Sankyo |
22677529 |
3 |
Pyrrolidinobenzoic acid inhibitors of influenza virus neuraminidase: the hydrophobic side chain influences type A subtype selectivity. |
University of Alabama At Birmingham |
18694948 |
17 |
Limited inhibitory effects of oseltamivir and zanamivir on human sialidases. |
Miyagi Cancer Center Research Institute |
15214773 |
76 |
Fragment-based drug discovery. |
Sunesis Pharmaceuticals |
11000002 |
10 |
BCX-1812 (RWJ-270201): discovery of a novel, highly potent, orally active, and selective influenza neuraminidase inhibitor through structure-based drug design. |
Biocryst Pharmaceuticals |
10602699 |
15 |
Binding constants of neuraminidase inhibitors: An investigation of the linear interaction energy method. |
University of Southampton |
9526556 |
18 |
Dihydropyrancarboxamides related to zanamivir: a new series of inhibitors of influenza virus sialidases. 2. Crystallographic and molecular modeling study of complexes of 4-amino-4H-pyran-6-carboxamides and sialidase from influenza virus types A and B. |
Glaxo Wellcome Research and Development |
8126701 |
3 |
Molecular modeling studies on ligand binding to sialidase from influenza virus and the mechanism of catalysis. |
Monash University |
11266166 |
36 |
Sialidase inhibitors related to zanamivir. Further SAR studies of 4-amino-4H-pyran-2-carboxylic acid-6-propylamides. |
Glaxowellcome Medicines Research Centre |
| 22 |
Novel inhibitors of influenza sialidases related to zanamivir. Heterocyclic replacements of the glycerol sidechain |
TBA |
| 51 |
Novel inhibitors of influenza sialidases related to GG167 structure-activity, crystallographic and Molecular dynamics studies with 4H-pyran-2-carboxylic acid 6-carboxamides |
TBA |
| 16 |
Novel inhibitors of influenza sialidase related to GG167 Synthesis of 4-amino and guanidino-4H-pyran-2-carboxylic acid-6-propylamides; selective inhibitors of influenza a virus sialidase |
TBA |
22100261 |
12 |
Synthesis and biological evaluation of sialic acid derivatives containing a long hydrophobic chain at the anomeric position and their C-5 linked polymers as potent influenza virus inhibitors. |
Saitama University |
21843936 |
35 |
3D QSAR and docking study of flavone derivatives as potent inhibitors of influenza H1N1 virus neuraminidase. |
Chinese Academy of Medical Sciences |
20014777 |
6 |
Antiviral potential and molecular insight into neuraminidase inhibiting diarylheptanoids from Alpinia katsumadai. |
University of Innsbruck |
15828835 |
6 |
Dimeric zanamivir conjugates with various linking groups are potent, long-lasting inhibitors of influenza neuraminidase including H5N1 avian influenza. |
Glaxosmithkline |
15582424 |
6 |
Design, synthesis, and structural analysis of inhibitors of influenza neuraminidase containing a 2,3-disubstituted tetrahydrofuran-5-carboxylic acid core. |
Abbott Laboratories |
11312919 |
22 |
Design, synthesis, and structural analysis of influenza neuraminidase inhibitors containing pyrrolidine cores. |
Abbott Laboratories |
31744778 |
11 |
Design, synthesis and biological evaluation of substituted flavones and aurones as potential anti-influenza agents. |
Prin. K.M. Kundnani College of Pharmacy |
30576902 |
36 |
Boronate, trifluoroborate, sulfone, sulfinate and sulfonate congeners of oseltamivir carboxylic acid: Synthesis and anti-influenza activity. |
National Taiwan University |
31835169 |
68 |
Discovery of novel 1,2,3-triazole oseltamivir derivatives as potent influenza neuraminidase inhibitors targeting the 430-cavity. |
Shandong University |
10395473 |
19 |
Potent inhibition of influenza sialidase by a benzoic acid containing a 2-pyrrolidinone substituent. |
University of Alabama At Birmingham |
31324565 |
12 |
Total synthesis of dryocrassin ABBA and its analogues with potential inhibitory activity against drug-resistant neuraminidases. |
Chinese Academy of Sciences |
31176096 |
44 |
Design, synthesis and biological evaluation of "Multi-Site"-binding influenza virus neuraminidase inhibitors. |
Shandong University |
31128993 |
22 |
Investigation of flexibility of neuraminidase 150-loop using tamiflu derivatives in influenza A viruses H1N1 and H5N1. |
Charles University |
31857844 |
1 |
Discovery of Novel Neuraminidase Inhibitors by Structure-Based Virtual Screening, Structural Optimization, and Bioassay. |
Shanghai Institute of Technology |
31708183 |
3 |
Design, synthesis and biological evaluation of oseltamivir derivatives containing pyridyl group as potent inhibitors of neuraminidase for influenza A. |
Wuyi University |
23411074 |
2 |
Aspulvinones from a mangrove rhizosphere soil-derived fungus Aspergillus terreus Gwq-48 with anti-influenza A viral (H1N1) activity. |
Ocean University of China |
20116898 |
52 |
QSAR study of flavonoids and biflavonoids as influenza H1N1 virus neuraminidase inhibitors. |
Universidad De Buenos Aires |
29107426 |
16 |
Synthesis and biological evaluation of NH |
Shenyang Pharmaceutical University |
29198893 |
3 |
Synthesis and anti-influenza virus evaluation of triterpene-sialic acid conjugates. |
Meiji Pharmaceutical University |
28958846 |
24 |
Discovery of berberine based derivatives as anti-influenza agent through blocking of neuraminidase. |
Konkuk University |
29965752 |
158 |
Optimization of N-Substituted Oseltamivir Derivatives as Potent Inhibitors of Group-1 and -2 Influenza A Neuraminidases, Including a Drug-Resistant Variant. |
Shandong University |
28984452 |
6 |
C-Methylated Flavonoid Glycosides from Pentarhizidium orientale Rhizomes and Their Inhibitory Effects on the H1N1 Influenza Virus. |
Seoul National University |
16621549 |
40 |
Novel 5-azaindole factor VIIa inhibitors. |
Celera |
14561087 |
27 |
Structure-activity relationships of the p38alpha MAP kinase inhibitor 1-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)naph- thalen-1-yl]urea (BIRB 796). |
Boehringer Ingelheim Pharmaceuticals |
11896401 |
3 |
Inhibition of p38 MAP kinase by utilizing a novel allosteric binding site. |
Boehringer Ingelheim Pharmaceuticals |
15857116 |
5 |
1-(5-Chloro-2-alkoxyphenyl)-3-(5-cyanopyrazin-2-yl)ureas [correction of cyanopyrazi] as potent and selective inhibitors of Chk1 kinase: synthesis, preliminary SAR, and biological activities. |
Abbott Laboratories |
16303309 |
31 |
Bicyclic and tricyclic thiophenes as protein tyrosine phosphatase 1B inhibitors. |
Wyeth Research |
10694412 |
15 |
Thermodynamics of substrate binding to the chaperone SecB. |
Indian Institute of Science |