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29 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28435528 24 Discovery of Highly Selective Inhibitors of the Immunoproteasome Low Molecular Mass Polypeptide 2 (LMP2) Subunit.EBI Kezar Life Sciences
25006746 85 Structure-based design of฿1i or฿5i specific inhibitors of human immunoproteasomes.EBI Leiden Institute of Chemistry and Netherlands Proteomics Centre
24900849 17 Oxathiazolones Selectively Inhibit the Human Immunoproteasome over the Constitutive Proteasome.EBI Weill Cornell Medical College
24524217 65 Structurally novel highly potent proteasome inhibitors created by the structure-based hybridization of nonpeptidic belactosin derivatives and peptide boronates.EBI Hokkaido University
22978849 13 Molecular mechanisms of acquired proteasome inhibitor resistance.EBI University of California San Diego
19348473 12 Design and synthesis of an orally bioavailable and selective peptide epoxyketone proteasome inhibitor (PR-047).EBI Proteolix
32189500 56 LMP2 Inhibitors as a Potential Treatment for Alzheimer's Disease.EBI University of Kentucky
30639896 42 Covalent docking modelling-based discovery of tripeptidyl epoxyketone proteasome inhibitors composed of aliphatic-heterocycles.EBI Hangzhou Institute of Innovative Medicine
31560200 30 Selective Phenylimidazole-Based Inhibitors of the EBI Weill Cornell Medicine
30611983 48 Exploration of novel macrocyclic dipeptide N-benzyl amides as proteasome inhibitors.EBI Zhejiang University
30380863 196 Required Immunoproteasome Subunit Inhibition Profile for Anti-Inflammatory Efficacy and Clinical Candidate KZR-616 ((2 S,3 R)- N-(( S)-3-(Cyclopent-1-en-1-yl)-1-(( R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-hydroxy-3-(4-methoxyphenyl)-2-(( S)-2-(2-morpholinoacetamido)propanamido)propenamide).EBI Kezar Life Sciences
31521028 67 Immunoproteasome-selective inhibitors: An overview of recent developments as potential drugs for hematologic malignancies and autoimmune diseases.EBI Hangzhou Xixi Hospital
30657666 263 Structure-Based Design of Inhibitors Selective for Human Proteasome ?2c or ?2i Subunits.EBI Leiden Institute of Chemistry and Netherlands Proteomics Centre
31177777 54 Improvement of Asparagine Ethylenediamines as Anti-malarial EBI Weill Cornell Medicine
31670954 9 The Immunoproteasome: An Emerging Target in Cancer and Autoimmune and Neurological Disorders.EBI Purdue University
30391816 43 Design, synthesis, and biological evaluation of novel phenol ether derivatives as non-covalent proteasome inhibitors.EBI Zhejiang University
30455150 10 Tetradehydrohalicyclamine B, a new proteasome inhibitor from the marine sponge Acanthostrongylophora ingens.EBI Kumamoto University
30165344 63 Design, synthesis, and evaluation of cystargolide-based ?-lactones as potent proteasome inhibitors.EBI New Mexico Institute of Mining and Technology
29339252 124 Structure-based design of human immuno- and constitutive proteasomes inhibitors.EBI Universit£
29782167 48 Potent and Highly Selective Inhibitors of the Proteasome Trypsin-like Site by Incorporation of Basic Side Chain Containing Amino Acid Derived Sulfonyl Fluorides.EBI University of Glasgow
2250662 140 Characterization of muscarinic M4 binding sites in rabbit lung, chicken heart, and NG108-15 cells.BDB Glaxo Group Research