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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
18242984 6 Constraining the amide bond in N-sulfonylated dipeptide VLA-4 antagonists.EBI Merck Research Laboratories
20705461 38 Synthesis and biological activity of N-substituted aminocarbonyl-1,3-dioxolanes as VLA-4 antagonists.EBI New Drug Discovery Research
20022493 35 Heterocycle-substituted proline dipeptides as potent VLA-4 antagonists.EBI Merck Research Laboratories
19441819 17 Discovery of N-{N-[(3-cyanophenyl)sulfonyl]-4(R)-cyclobutylamino-(L)-prolyl}-4-[(3',5'-dichloroisonicotinoyl) amino]-(L)-phenylalanine (MK-0668), an extremely potent and orally active antagonist of very late antigen-4.EBI Merck Research Laboratories
19124247 9 A novel and potent VLA-4 antagonist based on trans-4-substituted cyclohexanecarboxylic acid.EBI Daiichi Sankyo
19072684 11 Selectively targeting T- and B-cell lymphomas: a benzothiazole antagonist of alpha4beta1 integrin.EBI University of California Davis
18952443 26 Identification of 4-[1-[3-chloro-4-[N'-(5-fluoro-2-methylphenyl)ureido]phenylacetyl]-(4S)-fluoro-(2S)-pyrrolidinylmethoxy]benzoic acid as a potent, orally active VLA-4 antagonist.EBI Daiichi Sankyo
18539454 47 Imidazopyridines as VLA-4 integrin antagonists.EBI Ucb Pharma
18160288 31 Synthetic study of VLA-4/VCAM-1 inhibitors: synthesis and structure-activity relationship of piperazinylphenylalanine derivatives.EBI Kyowa Hakko Kogyo
10866374 11 The design and synthesis of potent cyclic peptide VCAM-VLA-4 antagonists incorporating an achiral Asp-Pro mimetic.EBI Roche Research Center
10866373 8 Cyclic thioether peptide mimetics as VCAM-VLA-4 antagonists.EBI Roche Research Center
10866372 7 Carbacyclic peptide mimetics as VCAM-VLA-4 antagonists.EBI Roche Research Center
23899692 10 Discovery of a potent and selective DDR1 receptor tyrosine kinase inhibitor.BDB Massachusetts General Hospital and Harvard Medical School