The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
19800231 |
92 |
Tetrahydroquinoline sulfonamides as vasopressin 1b receptor antagonists. |
Schering-Plough Research Institute |
17300166 |
88 |
Design and synthesis of the first selective agonists for the rat vasopressin V(1b) receptor: based on modifications of deamino-[Cys1]arginine vasopressin at positions 4 and 8. |
University of Montpellier |
10201826 |
24 |
Synthesis of oxytocin antagonists containing conformationally constrained amino acids in position 2. |
Albert Szent-Gy£Rgyi Medical University |
21353540 |
55 |
Synthesis and SAR studies of novel 2-(4-oxo-2-aryl-quinazolin-3(4H)-yl)acetamide vasopressin V1b receptor antagonists. |
Msd |
20550119 |
96 |
Oral oxytocin antagonists. |
Drugmoldesign |
20719508 |
26 |
Identification and optimization of novel 2-(4-oxo-2-aryl-quinazolin-3(4H)-yl)acetamide vasopressin V3 (V1b) receptor antagonists. |
Ligand Pharmaceuticals |
| 4 |
Vasopressin trisulphide: synthesis, NMR study and affinity studies with V1 and V2 subtypes receptors |
TBA |
14695824 |
68 |
Synthesis and structure-activity relationships of 5,6,7,8-tetrahydro-4H-thieno[3,2-b]azepine derivatives: novel arginine vasopressin antagonists. |
Central Pharmaceutical Research Institute |
12502367 |
17 |
New benzo[h][1,6]naphthyridine and azepino[3,2-c]quinoline derivatives as selective antagonists of 5-HT4 receptors: binding profile and pharmacological characterization. |
Université |
8258821 |
491 |
Nanomolar-affinity, non-peptide oxytocin receptor antagonists. |
Merck Research Laboratories |
30199637 |
172 |
LIT-001, the First Nonpeptide Oxytocin Receptor Agonist that Improves Social Interaction in a Mouse Model of Autism. |
Umr7200 Cnrs/Universit£ |
2416923 |
40 |
Arginine-vasopressin analogues with high antidiuretic/vasopressor selectivity. Synthesis, biological activity, and receptor binding affinity of arginine-vasopressin analogues with substitutions in positions 1, 2, 4, 7, and 8. |
TBA |
2163451 |
45 |
Cyclic hexapeptide oxytocin antagonists. Potency-, selectivity-, and solubility-enhancing modifications. |
Merck Sharp & Dohme Research Laboratories |
1331449 |
268 |
Orally active, nonpeptide oxytocin antagonists. |
Merck Research Laboratories |