BindingDB logo
myBDB logout

7 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
10201826 24 Synthesis of oxytocin antagonists containing conformationally constrained amino acids in position 2.EBI Albert Szent-Gy£Rgyi Medical University
 4 Vasopressin trisulphide: synthesis, NMR study and affinity studies with V1 and V2 subtypes receptorsEBI TBA
14695824 68 Synthesis and structure-activity relationships of 5,6,7,8-tetrahydro-4H-thieno[3,2-b]azepine derivatives: novel arginine vasopressin antagonists.EBI Central Pharmaceutical Research Institute
8258821 491 Nanomolar-affinity, non-peptide oxytocin receptor antagonists.EBI Merck Research Laboratories
2416923 40 Arginine-vasopressin analogues with high antidiuretic/vasopressor selectivity. Synthesis, biological activity, and receptor binding affinity of arginine-vasopressin analogues with substitutions in positions 1, 2, 4, 7, and 8.EBI TBA
2163451 45 Cyclic hexapeptide oxytocin antagonists. Potency-, selectivity-, and solubility-enhancing modifications.EBI Merck Sharp & Dohme Research Laboratories
1331449 268 Orally active, nonpeptide oxytocin antagonists.EBI Merck Research Laboratories