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35 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
7837233 21 CCK-A receptor selective antagonists derived from the CCK-A receptor selective tetrapeptide agonist Boc-Trp-Lys(Tac)-Asp-MePhe-NH2 (A-71623).EBI Glaxo Research Institute
9057851 30 Structure-based design of new constrained cyclic agonists of the cholecystokinin CCK-B receptor.EBI University of Paris
8831778 22 The use of topographical constraints in receptor mapping: investigation of the topographical requirements of the tryptophan 30 residue for receptor binding of Asp-Tyr-D-Phe-Gly-Trp-(N-Me)Nle-Asp-Phe-NH2 (SNF 9007), a cholecystokinin (26-33) analogue that binds to both CCK-B and delta-opioid receptoEBI University of Arizona
8126703 29 Tetrapeptide CCK-A agonists: effect of backbone N-methylations on in vitro and in vivo CCK activity.EBI Abbott Laboratories
8295219 44 Tetrapeptide CCK agonists: structure-activity studies on modifications at the N-terminus.EBI Abbott Laboratories
8201591 2 CCK-A-selective tetrapeptides containing lys(N epsilon)-amide residues: favorable in vivo and in vitro effects of N-methylation at the aspartyl residue.EBI Abbott Laboratories
8421283 43 CCK-B agonist or antagonist activities of structurally hindered and peptidase-resistant Boc-CCK4 derivatives.EBI University of Paris
1375964 112 Development of potent and selective CCK-A receptor agonists from Boc-CCK-4: tetrapeptides containing Lys(N epsilon)-amide residues.EBI Abbott Laboratories
2299627 54 Novel glutamic acid derived cholecystokinin receptor ligands.EBI Merck Sharp & Dohme Research Laboratories
1700123 26 Development of CCK-tetrapeptide analogues as potent and selective CCK-A receptor agonists.EBI Abbott Laboratories
2885419 179 Design of nonpeptidal ligands for a peptide receptor: cholecystokinin antagonists.EBI TBA
14698161 10 Synthesis and biological characterisation of [3H]BBL454, a new CCK2 selective radiolabelled agonist displaying original pharmacological properties.EBI University of Paris
 32 Pseudopeptide CCK-4 analogues incorporating the [CH(CN)NH] peptide bond surrogateEBI TBA
 66 Amino acid-derived piperidides as novel CCKB ligands with anxiolytic-like propertiesEBI TBA
 42 A water soluble benzazepine cholecystokinin-B receptor antagonistEBI TBA
 58 5,7-Diphenyl-3-ureidohexahydroazepin-2-ones as Cholecystokinin-B receptor ligandsEBI TBA
 28 Toward developing peptidomimetics: Successful replacement of backbone amide bonds in tetrapeptide-based CCK-A receptor agonistsEBI TBA
 16 Structure-based design and pharmacological properties of potent selective and systemically active CCK-B peptidomimeticsEBI TBA
19261479 21 Anthranilic acid based CCK1 receptor antagonists: blocking the receptor with the same 'words' of the endogenous ligand.EBI University of Trieste
17368898 6 Synthesis and evaluation of novel benzimidazole derivative [Bz-Im] and its radio/biological studies.EBI Lucknow University
11020275 75 Replacement of glycine with dicarbonyl and related moieties in analogues of the C-terminal pentapeptide of cholecystokinin: CCK(2) agonists displaying a novel binding mode.EBI University of Paris
9871777 28 Novel constrained CCK-B dipeptoid antagonists derived from pipecolic acid.EBI University of Paris
9089338 29 Minor structural differences in Boc-CCK-4 derivatives dictate affinity and selectivity for CCK-A and CCK-B receptors.EBI Abbott Laboratories
8411002 67 Cholecystokinin peptidomimetics as selective CCK-B antagonists: design, synthesis, and in vitro and in vivo biochemical properties.EBI University of Paris
8201590 20 Novel Asp32-replacement tetrapeptide analogues as potent and selective CCK-A agonists.EBI Abbott Laboratories
7966138 55 5-Phenyl-3-ureidobenzazepin-2-ones as cholecystokinin-B receptor antagonists.EBI Pfizer
2724293 28 Synthesis and binding affinities of cyclic and related linear analogues of CCK8 selective for central receptors.EBI University of Paris
2704023 20 Hybrid cholecystokinin (CCK) antagonists: new implications in the design and modification of CCK antagonists.EBI Abbott Laboratories
2464062 10 Full agonists of CCK8 containing a nonhydrolyzable sulfated tyrosine residue.EBI University of Paris
1992147 10 trans-3-n-propyl-L-proline is a highly favorable, conformationally restricted replacement for methionine in the C-terminal tetrapeptide of cholecystokinin. Stereoselective synthesis of 3-allyl- and 3-n-propyl-L-proline derivatives from 4-hydroxy-L-proline.EBI Abbott Laboratories
1766000 90 Cholecystokinin antagonists: (R)-tryptophan-based hybrid antagonists of high affinity and selectivity for CCK-A receptors.EBI Abbott Laboratories
1716682 64 Boc-CCK-4 derivatives containing side-chain ureas as potent and selective CCK-a receptor agonists.EBI Abbott Laboratories
1701834 20 Boc-Trp-Orn(Z)-Asp-NH2 and derivatives: a new family of CCK antagonists.EBI University of Paris
1501220 52 Synthesis and biological activity of CCK heptapeptide analogues. Effects of conformational constraints and standard modifications on receptor subtype selectivity, functional activity in vitro, and appetite suppression in vivo.EBI Abbott Laboratories
1495013 24 N-methylated analogs of Ac[Nle28,31]CCK(26-33): synthesis, activity, and receptor selectivity.EBI Hadassah-University Hospital