The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
7837233 |
21 |
CCK-A receptor selective antagonists derived from the CCK-A receptor selective tetrapeptide agonist Boc-Trp-Lys(Tac)-Asp-MePhe-NH2 (A-71623). |
Glaxo Research Institute |
9057851 |
30 |
Structure-based design of new constrained cyclic agonists of the cholecystokinin CCK-B receptor. |
University of Paris |
8831778 |
22 |
The use of topographical constraints in receptor mapping: investigation of the topographical requirements of the tryptophan 30 residue for receptor binding of Asp-Tyr-D-Phe-Gly-Trp-(N-Me)Nle-Asp-Phe-NH2 (SNF 9007), a cholecystokinin (26-33) analogue that binds to both CCK-B and delta-opioid recepto |
University of Arizona |
8126703 |
29 |
Tetrapeptide CCK-A agonists: effect of backbone N-methylations on in vitro and in vivo CCK activity. |
Abbott Laboratories |
8295219 |
44 |
Tetrapeptide CCK agonists: structure-activity studies on modifications at the N-terminus. |
Abbott Laboratories |
8201591 |
2 |
CCK-A-selective tetrapeptides containing lys(N epsilon)-amide residues: favorable in vivo and in vitro effects of N-methylation at the aspartyl residue. |
Abbott Laboratories |
8421283 |
43 |
CCK-B agonist or antagonist activities of structurally hindered and peptidase-resistant Boc-CCK4 derivatives. |
University of Paris |
1375964 |
112 |
Development of potent and selective CCK-A receptor agonists from Boc-CCK-4: tetrapeptides containing Lys(N epsilon)-amide residues. |
Abbott Laboratories |
2299627 |
54 |
Novel glutamic acid derived cholecystokinin receptor ligands. |
Merck Sharp & Dohme Research Laboratories |
1700123 |
26 |
Development of CCK-tetrapeptide analogues as potent and selective CCK-A receptor agonists. |
Abbott Laboratories |
2885419 |
179 |
Design of nonpeptidal ligands for a peptide receptor: cholecystokinin antagonists. |
TBA |
14698161 |
10 |
Synthesis and biological characterisation of [3H]BBL454, a new CCK2 selective radiolabelled agonist displaying original pharmacological properties. |
University of Paris |
| 32 |
Pseudopeptide CCK-4 analogues incorporating the [CH(CN)NH] peptide bond surrogate |
TBA |
| 66 |
Amino acid-derived piperidides as novel CCKB ligands with anxiolytic-like properties |
TBA |
| 42 |
A water soluble benzazepine cholecystokinin-B receptor antagonist |
TBA |
| 58 |
5,7-Diphenyl-3-ureidohexahydroazepin-2-ones as Cholecystokinin-B receptor ligands |
TBA |
| 28 |
Toward developing peptidomimetics: Successful replacement of backbone amide bonds in tetrapeptide-based CCK-A receptor agonists |
TBA |
| 16 |
Structure-based design and pharmacological properties of potent selective and systemically active CCK-B peptidomimetics |
TBA |
19261479 |
21 |
Anthranilic acid based CCK1 receptor antagonists: blocking the receptor with the same 'words' of the endogenous ligand. |
University of Trieste |
17368898 |
6 |
Synthesis and evaluation of novel benzimidazole derivative [Bz-Im] and its radio/biological studies. |
Lucknow University |
11020275 |
75 |
Replacement of glycine with dicarbonyl and related moieties in analogues of the C-terminal pentapeptide of cholecystokinin: CCK(2) agonists displaying a novel binding mode. |
University of Paris |
9871777 |
28 |
Novel constrained CCK-B dipeptoid antagonists derived from pipecolic acid. |
University of Paris |
9089338 |
29 |
Minor structural differences in Boc-CCK-4 derivatives dictate affinity and selectivity for CCK-A and CCK-B receptors. |
Abbott Laboratories |
8411002 |
67 |
Cholecystokinin peptidomimetics as selective CCK-B antagonists: design, synthesis, and in vitro and in vivo biochemical properties. |
University of Paris |
8201590 |
20 |
Novel Asp32-replacement tetrapeptide analogues as potent and selective CCK-A agonists. |
Abbott Laboratories |
7966138 |
55 |
5-Phenyl-3-ureidobenzazepin-2-ones as cholecystokinin-B receptor antagonists. |
Pfizer |
2724293 |
28 |
Synthesis and binding affinities of cyclic and related linear analogues of CCK8 selective for central receptors. |
University of Paris |
2704023 |
20 |
Hybrid cholecystokinin (CCK) antagonists: new implications in the design and modification of CCK antagonists. |
Abbott Laboratories |
2464062 |
10 |
Full agonists of CCK8 containing a nonhydrolyzable sulfated tyrosine residue. |
University of Paris |
1992147 |
10 |
trans-3-n-propyl-L-proline is a highly favorable, conformationally restricted replacement for methionine in the C-terminal tetrapeptide of cholecystokinin. Stereoselective synthesis of 3-allyl- and 3-n-propyl-L-proline derivatives from 4-hydroxy-L-proline. |
Abbott Laboratories |
1766000 |
90 |
Cholecystokinin antagonists: (R)-tryptophan-based hybrid antagonists of high affinity and selectivity for CCK-A receptors. |
Abbott Laboratories |
1716682 |
64 |
Boc-CCK-4 derivatives containing side-chain ureas as potent and selective CCK-a receptor agonists. |
Abbott Laboratories |
1701834 |
20 |
Boc-Trp-Orn(Z)-Asp-NH2 and derivatives: a new family of CCK antagonists. |
University of Paris |
1501220 |
52 |
Synthesis and biological activity of CCK heptapeptide analogues. Effects of conformational constraints and standard modifications on receptor subtype selectivity, functional activity in vitro, and appetite suppression in vivo. |
Abbott Laboratories |
1495013 |
24 |
N-methylated analogs of Ac[Nle28,31]CCK(26-33): synthesis, activity, and receptor selectivity. |
Hadassah-University Hospital |