The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
2477546 |
16 |
Synthesis and biological activity of some partially modified retro-inverso analogues of cholecystokinin. |
Centre De Pharmacologie-Endocrinologie (Montpellier, France) |
3336026 |
18 |
Cholecystokinin antagonists. Synthesis and biological evaluation of 3-substituted 1,4-benzodiazepin-2-amines. |
Merck Sharp & Dohme Research Laboratories |
2441054 |
18 |
Synthesis and biological activities of pseudopeptide analogues of the C-terminal heptapeptide of cholecystokinin. On the importance of the peptide bonds. |
TBA |
3761313 |
22 |
Cholecystokinin antagonists. Synthesis of asperlicin analogues with improved potency and water solubility. |
TBA |
2848124 |
401 |
Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists. |
Merck Sharp & Dohme Research Laboratories |
| 16 |
Conversion of acyclic nonpeptide CCK antagonists into CCK agonists |
Glaxo Wellcome Research and Development |
16722631 |
87 |
An integrated in silico 3D model-driven discovery of a novel, potent, and selective amidosulfonamide 5-HT1A agonist (PRX-00023) for the treatment of anxiety and depression. |
Predix Pharmaceuticals |
10377216 |
4 |
A peptide agonist acts by occupation of a monomeric G protein-coupled receptor: dual sites of covalent attachment to domains near TM1 and TM7 of the same molecule make biologically significant domain-swapped dimerization unlikely. |
Mayo Clinic and Foundation |
1501220 |
52 |
Synthesis and biological activity of CCK heptapeptide analogues. Effects of conformational constraints and standard modifications on receptor subtype selectivity, functional activity in vitro, and appetite suppression in vivo. |
Abbott Laboratories |
1495013 |
24 |
N-methylated analogs of Ac[Nle28,31]CCK(26-33): synthesis, activity, and receptor selectivity. |
Hadassah-University Hospital |