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22 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27654218 56 Synthesis and biological evaluation of a series of N-alkylated imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.EBI Ludwig-Maximilians-Universit£T M£Nchen
27039250 58 Synthesis of 4-substituted nipecotic acid derivatives and their evaluation as potential GABA uptake inhibitors.EBI Ludwig-Maximilians-Universit£T M£Nchen
26706177 136 Straightforward and effective synthesis of¿-aminobutyric acid transporter subtype 2-selective acyl-substituted azaspiro[4.5]decanes.EBI Universit£
25882526 496 Structure activity relationship of selective GABA uptake inhibitors.EBI University of Copenhagen
25025595 30 First photoswitchable neurotransmitter transporter inhibitor: light-induced control of¿-aminobutyric acid transporter 1 (GAT1) activity in mouse brain.EBI Ludwig-Maximilians-Universit£T M£Nchen
24973660 150 Synthesis, biological evaluation and structure-activity relationship of new GABA uptake inhibitors, derivatives of 4-aminobutanamides.EBI Jagiellonian University Medical College
23398473 85 Selective mGAT2 (BGT-1) GABA uptake inhibitors: design, synthesis, and pharmacological characterization.EBI University of Copenhagen
21940173 32 Aminomethyltetrazoles as potential inhibitors of the¿-aminobutyric acid transporters mGAT1-mGAT4: synthesis and biological evaluation.EBI Ludwig-Maximilians-University Munich
21353350 61 Development of imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.EBI Ludwig-Maximilians-University Munich
30718063 118 Synthesis and biological evaluation of novel N-substituted nipecotic acid derivatives with a cis-alkene spacer as GABA uptake inhibitors.EBI Ludwig-Maximilians-Universit£T M£Nchen
30777661 42 Screening oxime libraries by means of mass spectrometry (MS) binding assays: Identification of new highly potent inhibitors to optimized inhibitors ?-aminobutyric acid transporter 1.EBI Ludwig-Maximilians-University M£Nchen
30503411 15 Generation and screening of pseudostatic hydrazone libraries derived from 5-substituted nipecotic acid derivatives at the GABA transporter mGAT4.EBI Ludwig-Maximilians-Universit£T M£Nchen
30376325 50 Novel Allosteric Ligands of ?-Aminobutyric Acid Transporter 1 (GAT1) by MS Based Screening of Pseudostatic Hydrazone Libraries.EBI Ludwig-Maximilians-Universit£T M£Nchen
23859778 107 2-Substituted 4-hydroxybutanamides as potential inhibitors of ?-aminobutyric acid transporters mGAT1-mGAT4: synthesis and biological evaluation.EBI Jagiellonian University Medical College
23598250 49 Synthesis and evaluation of N-substituted nipecotic acid derivatives with an unsymmetrical bis-aromatic residue attached to a vinyl ether spacer as potential GABA uptake inhibitors.EBI Ludwig-Maximilians-University Munich
30442505 61 Synthesis and biological evaluation of novel N-substituted nipecotic acid derivatives with a trans-alkene spacer as potent GABA uptake inhibitors.EBI Ludwig-Maximilians-Universit£T M£Nchen
29924931 58 Development of New Photoswitchable Azobenzene Based ?-Aminobutyric Acid (GABA) Uptake Inhibitors with Distinctly Enhanced Potency upon Photoactivation.EBI Ludwig-Maximilians-University Munich
29886082 74 Synthesis and biological evaluation of novel N-substituted nipecotic acid derivatives with an alkyne spacer as GABA uptake inhibitors.EBI Ludwig-Maximilians-Universit£T M£Nchen
28991462 360 Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/?-Aminobutyric Acid Transporter 1 (BGT1).EBI University of Copenhagen