The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 26346669 |
53 |
Synthesis of new opioid derivatives with a propellane skeleton and their pharmacologies: Part 5, novel pentacyclic propellane derivatives with a 6-amide side chain. |
University of Tsukuba |
| 26252963 |
15 |
Novel diazabicycloalkane delta opioid agonists. |
Istituto Di Farmacologia Traslazionale |
| 25783191 |
87 |
Design, syntheses, and pharmacological characterization of 17-cyclopropylmethyl-3,14ß-dihydroxy-4,5a-epoxy-6a-(isoquinoline-3'-carboxamido)morphinan analogues as opioid receptor ligands. |
Virginia Commonwealth University |
| 23116891 |
15 |
Synthesis of new opioid derivatives with a propellane skeleton and their pharmacologies: part 3, novel propellane derivatives with pentacyclic skeletons. |
Kitasato University |
| 22734622 |
78 |
Synthesis and evaluation of aryl-naloxamide opiate analgesics targeting truncated exon 11-associatedµ opioid receptor (MOR-1) splice variants. |
Memorial Sloan-Kettering Cancer Center |
| 18829333 |
28 |
Design, synthesis, and structure-activity relationship of novel opioid kappa-agonists. |
Toray Industries |
| 17702750 |
1 |
Long-acting kappa opioid antagonists disrupt receptor signaling and produce noncompetitive effects by activating c-Jun N-terminal kinase. |
University of Washington |
| 9379438 |
31 |
Discovery of a novel class of substituted pyrrolooctahydroisoquinolines as potent and selective delta opioid agonists, based on an extension of the message-address concept. |
Smithkline Beecham |
| 9207938 |
15 |
Pyrrolomorphinans as delta opioid receptor antagonists. The role of steric hindrance in conferring selectivity. |
University of Minnesota |
| 9171881 |
17 |
7-Spiroindanyl derivatives of naltrexone and oxymorphone as selective ligands for delta opioid receptors. |
University of Minnesota |
| 8648612 |
30 |
Arylacetamide-derived fluorescent probes: synthesis, biological evaluation, and direct fluorescent labeling of kappa opioid receptors in mouse microglial cells. |
University of Minnesota |
| 2549247 |
39 |
Benzofuro[2,3-c]pyridin-6-ols: synthesis, affinity for opioid-receptor subtypes, and antinociceptive activity. |
Ciba-Geigy |
| | 36 |
Pyrrolooctahydroisoquinolines as potent and selective opioid receptor ligands: SAR analysis and docking studies |
TBA |
| 21392859 |
1 |
Synthesis and biological evaluation of dibenz[b,f][1,5]oxazocine derivatives for agonist activity at κ-opioid receptor. |
Indian Institute of Chemical Biology |
| | 26 |
6N-Cinnamoyl-β-naltrexamine and its p-nitro derivative. High efficacy κ-opioid agonists with weak antagonist actions |
TBA |
| 12408719 |
21 |
Synthesis and structure-activity relationships of an orally available and long-acting analgesic peptide, N(alpha)-amidino-Tyr-D-Arg-Phe-MebetaAla-OH (ADAMB). |
Daiichi Fine Chemical |
| 11150174 |
84 |
Synthesis and in vitro and in vivo activity of (-)-(1R,5R,9R)- and (+)-(1S,5S,9S)-N-alkenyl-, -N-alkynyl-, and -N-cyanoalkyl-5, 9-dimethyl-2'-hydroxy-6,7-benzomorphan homologues. |
Virginia Commonwealth University |
| 27556704 |
64 |
Mitragynine/Corynantheidine Pseudoindoxyls As Opioid Analgesics with Mu Agonism and Delta Antagonism, Which Do Not Recruit ?-Arrestin-2. |
Memorial Sloan Kettering Cancer Center |
| 30608693 |
48 |
Design, Synthesis, and Biological Evaluation of the Third Generation 17-Cyclopropylmethyl-3,14?-dihydroxy-4,5?-epoxy-6?-[(4'-pyridyl)carboxamido]morphinan (NAP) Derivatives as ?/? Opioid Receptor Dual Selective Ligands. |
Virginia Commonwealth University |
| 9301669 |
24 |
7-spirobenzocyclohexyl derivatives of naltrexone, oxymorphone, and hydromorphone as selective opioid receptor ligands. |
University of Minnesota |
| 31782922 |
107 |
Application of Bivalent Bioisostere Concept on Design and Discovery of Potent Opioid Receptor Modulators. |
Virginia Commonwealth University |
| 24103580 |
36 |
Novel 6?-acylaminomorphinans with analgesic activity. |
Semmelweis University |
| 24090913 |
42 |
Synthesis and biological evaluation of novel delta (?) opioid receptor ligands with diazatricyclodecane skeletons. |
C.N.R. Istituto Di Farmacologia Traslazionale |
| 23948248 |
52 |
Structure activity relationship studies of 17-cyclopropylmethyl-3,14?-dihydroxy-4,5?-epoxy-6?-(isoquinoline-3'-carboxamido)morphinan (NAQ) analogues as potent opioid receptor ligands: preliminary results on the role of electronic characteristics for affinity and function. |
Virginia Commonwealth University |
| 23880538 |
51 |
Access to 7?-analogs of codeine with mixed ?/? agonist activity via 6,7-?-epoxide opening. |
University of Texas At Austin |
| 7932577 |
24 |
Selective kappa-opioid agonists: synthesis and structure-activity relationships of piperidines incorporating on oxo-containing acyl group. |
Smithkline Beecham Farmaceutici |
| 1967312 |
91 |
Synthesis and structure-activity relationships of dynorphin A-(1-8) amide analogues. |
Eisai |
| 1648141 |
21 |
Naphtho and benzo analogues of the kappa opioid agonist trans-(+/-)-3,4-dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl] benzeneacetamide. |
University of Notre Dame |
| 26520885 |
21 |
Synthesis of 4-thiazolidinone analogs as potent in vitro anti-urease agents. |
Hazara University |
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