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The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28530802 121 Discovery of N-(5-Fluoropyridin-2-yl)-6-methyl-4-(pyrimidin-5-yloxy)picolinamide (VU0424238): A Novel Negative Allosteric Modulator of Metabotropic Glutamate Receptor Subtype 5 Selected for Clinical Evaluation.EBI Vanderbilt University Institute of Imaging Science