The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27140209 |
18 |
Urotensin II((4-11)) Azasulfuryl Peptides: Synthesis and Biological Activity. |
Universit£ |
25984647 |
56 |
De Novo Conception of Small Molecule Modulators Based on Endogenous Peptide Ligands: Pyrrolodiazepin-2-one¿-Turn Mimics That Differentially Modulate Urotensin II Receptor-Mediated Vasoconstriction ex Vivo. |
Universit£ |
24992374 |
33 |
Lead optimization of P5U and urantide: discovery of novel potent ligands at the urotensin-II receptor. |
University of Naples&Quot;Federico Ii&Quot |
24251366 |
78 |
Development and pharmacological characterization of conformationally constrained urotensin II-related peptide agonists. |
Universit£ |
23453841 |
58 |
Deconstruction of sulfonamide inhibitors of the urotensin receptor (UT) and design and synthesis of benzylamine and benzylsulfone antagonists. |
Boehringer Ingelheim Pharmaceuticals |
19432421 |
31 |
New insight into the binding mode of peptide ligands at Urotensin-II receptor: structure-activity relationships study on P5U and urantide. |
University of Naples Federico Ii |
20043680 |
49 |
Urotensin-II receptor modulators as potential drugs. |
Johnson & Johnson Pharmaceutical Research & Development |
19731961 |
127 |
Nonpeptide urotensin-II receptor antagonists: a new ligand class based on piperazino-phthalimide and piperazino-isoindolinone subunits. |
Johnson & Johnson Pharmaceutical Research & Development |
17933531 |
24 |
Phenylpiperidine-benzoxazinones as urotensin-II receptor antagonists: synthesis, SAR, and in vivo assessment. |
Johnson & Johnson Pharmaceutical Research & Development |
30615452 |
47 |
Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides. |
University of Naples "Federico Ii |
12408704 |
3 |
Discovery of the first nonpeptide agonist of the GPR14/urotensin-II receptor: 3-(4-chlorophenyl)-3-(2- (dimethylamino)ethyl)isochroman-1-one (AC-7954). |
Acadia Pharmaceuticals |
30183282 |
59 |
Discovery of New Allosteric Modulators of the Urotensinergic System through Substitution of the Urotensin II-Related Peptide (URP) Phenylalanine Residue. |
Universit£ |
29131958 |
70 |
Design, Synthesis, and Biological Assessment of Biased Allosteric Modulation of the Urotensin II Receptor Using Achiral 1,3,4-Benzotriazepin-2-one Turn Mimics. |
Universit£ |
26804375 |
22 |
Synthesis of Novel Oxazolo[4,5-b]pyridine-2-one based 1,2,3-triazoles as Glycogen Synthase Kinase-3ß Inhibitors with Anti-inflammatory Potential. |
Hamdard University (Jamia Hamdard) |