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8 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
25901531 211 Structure-activity relationship in a purine-scaffold compound series with selectivity for the endoplasmic reticulum Hsp90 paralog Grp94.EBI Sloan-Kettering Institute For Cancer Research
23965125 26 Experimental and structural testing module to analyze paralogue-specificity and affinity in the Hsp90 inhibitors series.EBI Memorial Sloan-Kettering Cancer Center
16854066 44 Design, synthesis, and biological evaluation of hydroquinone derivatives of 17-amino-17-demethoxygeldanamycin as potent, water-soluble inhibitors of Hsp90.EBI Infinity Pharmaceuticals
30351001 16 Discovery of a Potent Grp94 Selective Inhibitor with Anti-Inflammatory Efficacy in a Mouse Model of Ulcerative Colitis.EBI China Pharmaceutical University
29057043 40 Resorcinol-Based Grp94-Selective Inhibitors.EBI The University of Kansas
29528635 14 Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding.EBI Hauptman-Woodward Medical Research Institute