The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
10386934 |
15 |
Dual-acting agents with alpha1-adrenoceptor antagonistic and steroid 5alpha-reductase inhibitory activities. Synthesis and evaluation of arylpiperazine derivatives. |
Zeria Pharmaceutical |
9873656 |
17 |
Synthesis of benzanilide derivatives as dual acting agents with alpha 1-adrenoceptor antagonistic action and steroid 5-alpha reductase inhibitory activity. |
Zeria Pharmaceutical |
9873464 |
6 |
A practical synthesis of 3-substituted delta 3,5(6)-steroids as new potential 5 alpha-reductase inhibitor. |
Chinese Academy of Science |
2308144 |
16 |
Steroidal A ring aryl carboxylic acids: a new class of steroid 5 alpha-reductase inhibitors. |
Smith Kline & French Laboratories |
12139451 |
41 |
Synthesis and evaluation of 2'-substituted 4-(4'-carboxy- or 4'-carboxymethylbenzylidene)-N-acylpiperidines: highly potent and in vivo active steroid 5alpha-reductase type 2 inhibitors. |
Saarland University |
9135028 |
114 |
Pharmacological options in the treatment of benign prostatic hyperplasia. |
Pfizer |
8978835 |
18 |
Indole derivatives as a new class of steroid 5 alpha-reductase inhibitors. |
Kyowa Hakko Kogyo |
7629802 |
48 |
Structure-activity relationships for inhibition of type 1 and 2 human 5 alpha-reductase and human adrenal 3 beta-hydroxy-delta 5-steroid dehydrogenase/3-keto-delta 5-steroid isomerase by 6-azaandrost-4-en-3-ones: optimization of the C17 substituent. |
Glaxo Inc. Research Institute |
3783591 |
225 |
Azasteroids: structure-activity relationships for inhibition of 5 alpha-reductase and of androgen receptor binding. |
TBA |
9871588 |
5 |
Structure activity relationship study of known inhibitors of the enzyme 5 alpha-reductase (5AR). |
Kingston University |
21515045 |
2 |
Synthesis and bioactivity of new Finasteride conjugate. |
Jilin University |
29400967 |
136 |
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design. |
Bristol-Myers Squibb |
9871560 |
17 |
Synthesis and 5 alpha-reductase inhibitory activities of benzofuran derivatives with a carbamoyl group. |
Sankyo |
11689062 |
8 |
Novel lead generation through hypothetical pharmacophore three-dimensional database searching: discovery of isoflavonoids as nonsteroidal inhibitors of rat 5 alpha-reductase. |
TBA |
7636849 |
52 |
(E)-4-(2-[[3-(indol-5-yl)-1-oxo-2-butenyl]amino]phenoxy)butyric acid derivatives: a new class of steroid 5 alpha-reductase inhibitors in the rat prostate. 1. |
Kyowa Hakko Kogyo |
2391687 |
16 |
Hydroxyperfluoroazobenzenes: novel inhibitors of enzymes of androgen biosynthesis. |
Institute of Cancer Research |
2308145 |
48 |
Inhibition of steroid 5 alpha-reductase by unsaturated 3-carboxysteroids. |
Smith Kline & French Laboratories |